Acta Chimica Sinica ›› 1963, Vol. 29 ›› Issue (4): 260-265.
CHOW CHI-TING, KYI ZU-YOONG
It was shown by Shaw and Woolley that in a series of closely related derivatives of serotonin, etherification of the phenolic hydroxyl and introduction of a methyl group in the 2-position favoured the anti-serotonin activity.In the present work, seven derivatives of 3-(β-aminoethyl)-5-β-droxy-berizofuran, an isosteric compound of serotonin, have been synthesized;each of them carries a methyl group on the 2-position and has its 5-hydroxy group methylated, the amino group on the side chain being free or substituted.
CHOW CHI-TING, KYI ZU-YOONG. SEROTONIN ANALOGUES——Ⅱ. THE SYNTHESIS OF 2-METHYL-3-(β-AMINOETHYL)-5-METHOXY-BENZOFURAN AND ITS N-SUBSTITUTED DERIVATIVES[J]. Acta Chimica Sinica, 1963, 29(4): 260-265.
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