Chin. J. Org. Chem. ›› 2005, Vol. 25 ›› Issue (02): 176-181. Previous Articles     Next Articles

Original Articles



  1. (中山大学化学与化学工程学院 广州 510275)
  • 收稿日期:2004-03-25 修回日期:2004-08-31 发布日期:2005-01-15
  • 通讯作者: 许遵乐

Synthesis of 2-Arylbenzo[b]furan Derivatives

PANG Ji-Yan,WANG Bo,CHEN Zhi-Peng,XU Zun-Le*   

  1. (Department of Applied Chemistry, School of Chemistry and Chemical Engineering,
    Sun Yat-Sen University, Guangzhou 510275)
  • Received:2004-03-25 Revised:2004-08-31 Published:2005-01-15
  • Contact: XU Zun-Le

2-Arylbenzo[b]furans were obtained via coupling reaction of the copper(I) arylacetylides with the phenylbromide, and then a series of derivatives were designed and synthesized by reduction, Vilsmeier, hydrolysis and substituted reaction. All the compounds were fully characterized by MS, 1H NMR, IR spectra and elemental analysis.

Key words: synthesis, 2-benzo[b]furans, copper(I) arylacetylides