Chinese Journal of Organic Chemistry ›› 2021, Vol. 41 ›› Issue (10): 4007-4013.DOI: 10.6023/cjoc202105050 Previous Articles     Next Articles



芦军, 梁仁校, 贾义霞*()   

  1. 浙江工业大学化工学院 杭州 310014
  • 收稿日期:2021-05-29 修回日期:2021-07-31 发布日期:2021-08-17
  • 通讯作者: 贾义霞
  • 基金资助:
    国家自然科学基金(21702184); 国家自然科学基金(22071217); 国家自然科学基金(91956117)

Copper-Catalyzed Intramolecular Dearomative Arylation of Naphthylamines

Jun Lu, Renxiao Liang, Yixia Jia()   

  1. College of Chemical Engineering, Zhejiang University of Technology, Hangzhou 310014
  • Received:2021-05-29 Revised:2021-07-31 Published:2021-08-17
  • Contact: Yixia Jia
  • Supported by:
    National Natural Science Foundation of China(21702184); National Natural Science Foundation of China(22071217); National Natural Science Foundation of China(91956117)

A CuI-catalyzed intramolecular dearomative arylation of naphthylamines is developed through a Ullmann-type cross-coupling reaction, which led to a range of fused 3H-indole derivatives in good to excellent yields.

Key words: Ullmann coupling, naphthylamine, arylation, dearomatization