Chinese Journal of Organic Chemistry 2026, 46(1)

Please wait a minute...

- About the Cover:
  
  13 new thiochromone formamide derivatives substituted at position 2 were synthesized and two synthetic routes for these compounds were developed by Zhou, Su, Cui, Cheng, Li, Zhou, Sun, and Li on page 87. Their antifungal activities against Gaeumannomyces graminis/ var. tritici were evaluated in vitro by the plate method. The results of structure-activity relationship indicated that the group at position 2 of thiochromone formamide derivatives had an important influence on their antifungal activities against Gaeumannomyces graminis var. tritici.
- About the Cover:
  
  The nickel-catalyzed borylation of aryl nonaflates with B2pin2 is reported by Liang, Gui, Wang, Chu, Xu, and Shen on page 207. The reactions proceeded effectively via C—O bond cleavage to afford various valuable arylboronates in moderate to excellent yields with good functionality tolerance. Additionally, gram-scale synthesis and late-stage functionalization of aryl nonaflate derived from pterostilbene could also be realized.
2026, 46(1)

25 January 2026
Previous issue
Current Issue

REVIEWS ARTICLES HIGHLIGHTS

REVIEWS

Recent Advances on the Functionalization of Azlactones at Different Reactive Sites

Jiang Zhijie, Chen Jinxiu, Zhu Xiaofei, Deng Xinhao, Yan Qiongjiao, Wang Wei, Zhou Hui

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 1-20 DOI: 10.6023/cjoc202506007

Abstract( 73) HTML( 0) PDF(1112KB)( 28 )

Fig. & Tab. | References | Related Articles | Metrics

Recent Progress in the Total Synthesis of abeo-Steroids

Zhao Lilin, Li Zhaoqi, Zhong Liping, Min Long

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 21-38 DOI: 10.6023/cjoc202506022

Abstract( 146) HTML( 0) PDF(999KB)( 57 )

Fig. & Tab. | References | Related Articles | Metrics

Structural Modifications, Structure-Activity Relationships, and Total Synthesis Advances in Erythromycin Analogs against Resistant Pathogens

Cui Xinyi, Guo Lifan, Ma Congxuan, Li Yun, Liang Jianhua

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 39-73 DOI: 10.6023/cjoc202506020

Abstract( 56) HTML( 0) PDF(2154KB)( 22 )

Fig. & Tab. | References | Related Articles | Metrics

Progress in the Synthesis and Biological Studies of S-1-Propenyl-L-cysteine from Garlic

Tian Lingyan, Wang Shoufeng, Zeng Wei

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 74-86 DOI: 10.6023/cjoc202505028

Abstract( 44) HTML( 0) PDF(1498KB)( 10 )

Fig. & Tab. | References | Related Articles | Metrics

ARTICLES

Synthesis of Thiochromone Formamide Derivatives and Their Antifungal Activities

Zhou Pu, Su Ziyang, Cui Deyun, Cheng Yi-Nan, Li Yi, Zhou Haifeng, Sun Bingjian, Li Honglian

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 87-95 DOI: 10.6023/cjoc202506027

Abstract( 97) HTML( 0) PDF(675KB)( 109 )

Fig. & Tab. | References | Supporting Info. | Related Articles | Metrics

Study on the Cyclopropanation Reactivity and Selectivity of Spiroannulated Pentacyclic Diastereoisomers toward Synthesizing Cryptoquinonemethides

Zhang Yuanhe, Shen Yunjie, Tan Dongxing, Han Fushe

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 96-105 DOI: 10.6023/cjoc202508010

Abstract( 37) HTML( 0) PDF(774KB)( 15 )

Fig. & Tab. | References | Supporting Info. | Related Articles | Metrics

Study on the Synthesis and Fungicidal Activity of 1-Azolyl-1,1- diarylmethanes Containing Pyridine Ring

Hong Sai, Yin Fahong, Chen Minghui, Fu Bin, Xiao Yumei, Qin Zhaohai

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 106-117 DOI: 10.6023/cjoc202506035

Abstract( 97) HTML( 0) PDF(6147KB)( 59 )

Fig. & Tab. | References | Supporting Info. | Related Articles | Metrics

Silver-Catalyzed Tandem Decarboxylative Cyclization of 2,2-Difluoro-2-(phenylthio)acetic Acids with 2-Aryl-N-acrylamide Indoles

Liu Jiale, Tang Yucai, Yin Qiumei, Huang Jiaming, Deng Shiqiang, Xia Weiming, Jiang Jie, Wang Zu-Li

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 118-127 DOI: 10.6023/cjoc202507011

Abstract( 82) HTML( 0) PDF(537KB)( 33 )

Fig. & Tab. | References | Supporting Info. | Related Articles | Metrics

Synthesis and Characterization of Silacyclopropenes

Chen Yilin, Yue Jiayi, Lin Yiming, Liu Bingni, Dai Wen, Zhu Hongping

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 128-134 DOI: 10.6023/cjoc202506023

Abstract( 56) HTML( 0) PDF(1618KB)( 11 )

Fig. & Tab. | References | Supporting Info. | Related Articles | Metrics

Visible-Light-Driven Halogen-Bond-Induced Direct Coupling of Diethyl α-Iodomethylphosphonates with Coumarins/Quinolinones

Liang Jiarui, Li Jinlan, Jiang Yun, Yao Qiuli, Xu Yingshu, Wang Anjun

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 135-145 DOI: 10.6023/cjoc202506016

Abstract( 140) HTML( 0) PDF(1713KB)( 53 )

Fig. & Tab. | References | Supporting Info. | Related Articles | Metrics

Regio-reversed [3＋2] Cycloaddition of Triketone Enones with Nitrones

Han Tianjiao, Shi Qianqian, Fu Yundong, Mei Guangjian

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 146-155 DOI: 10.6023/cjoc202507022

Abstract( 51) HTML( 0) PDF(814KB)( 20 )

Fig. & Tab. | References | Supporting Info. | Related Articles | Metrics

Heterogeneous Copper Catalyzed Aerobic Oxidative Cross-Coupling of Tertiary Amines with Alkynes

Tan Ziyun, Yang Xin, Gong Shaofeng, Yang Huiling, Xie Yongyan, Zhang Jingya, Feng Zhetai, Li Wenyi, Xiao Xinsheng

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 156-166 DOI: 10.6023/cjoc202504020

Abstract( 102) HTML( 0) PDF(3132KB)( 56 )

Fig. & Tab. | References | Supporting Info. | Related Articles | Metrics

Copper-Catalyzed Asymmetric Oxidative Homocoupling Reaction of 3-Hydroxy-2-naphthoates: Design and Optimization of Amino Acid-Based Ligands

Wang Wen-Long, Wen Jia-Xu, Chen Fei, Bo Chunbo, Li Min, Liu Ning, Du Zhi-Hong

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 167-180 DOI: 10.6023/cjoc202505013

Abstract( 80) HTML( 0) PDF(2236KB)( 36 )

Fig. & Tab. | References | Supporting Info. | Related Articles | Metrics

Four-Component Hydroxythiolation of Styrenes with Imidazopyridines and Potassium Thiocyanate

Wang Yu, Huang Hongkun, Ling Chun, Chen Tian, Yao Hua, Yan Zhaohua

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 181-188 DOI: 10.6023/cjoc202506001

Abstract( 107) HTML( 0) PDF(458KB)( 54 )

Fig. & Tab. | References | Supporting Info. | Related Articles | Metrics

S-Heteroarylation of Cysteines

Zhang Xin, Li Fei, Zhou Chenxing, Huo Congde

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 189-198 DOI: 10.6023/cjoc202506011

Abstract( 95) HTML( 0) PDF(607KB)( 41 )

Fig. & Tab. | References | Supporting Info. | Related Articles | Metrics

Study on FeCl₃-Mediated Reaction of Aryl Boronic Esters with Electrophiles

Cui Lihua, Li Yatong, Wang Qifeng

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 199-206 DOI: 10.6023/cjoc202506018

Abstract( 66) HTML( 0) PDF(499KB)( 25 )

Fig. & Tab. | References | Supporting Info. | Related Articles | Metrics

Nickel-Catalyzed Borylation of Aryl Nonaflates for the Efficient Synthesis of Arylboronates via C—O Bond Functionalization

Liang Yuan, Gui Chao, Wang Wenwen, Chu Xueqiang, Xu Hao, Shen Zhiliang

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 207-214 DOI: 10.6023/cjoc202507010

Abstract( 87) HTML( 0) PDF(458KB)( 44 )

Fig. & Tab. | References | Supporting Info. | Related Articles | Metrics

Photocatalytic Radical-Mediated Synthesis of Unnatural α-Amino Acids from Heteroaryl Aldehydes

Ren Ke, Zhang Guanglu, Niu Yifan, Wang Xiaomeng, Chen Canyu, Jiang Min

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 215-224 DOI: 10.6023/cjoc202507030

Abstract( 116) HTML( 0) PDF(701KB)( 71 )

Fig. & Tab. | References | Supporting Info. | Related Articles | Metrics

PPh₃-Mediated One-Pot Synthesis of Indolin-3-ones from 2-Alkynylnitrobenzenes and Indoles

Feng Faxiu, Xu Shijie, Wang Xue, Yang Zhuoran, Wang Wenjun, Huang Shenlin, Zhang Xiaoxiang

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 225-232 DOI: 10.6023/cjoc202506013

Abstract( 122) HTML( 0) PDF(633KB)( 80 )

Fig. & Tab. | References | Supporting Info. | Related Articles | Metrics

Schiff Base Type Fe(III) Complexes Catalyzed Carbon Dioxide and Epoxides for Preparing Cyclic Carbonates

Liu Tao, Zhou Yongbo, Lang Tongqing, Niu Haibo, Chen Fei, Du Zhihong, Bo Chunbo, Li Min, Liu Ning

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 233-240 DOI: 10.6023/cjoc202506003

Abstract( 128) HTML( 0) PDF(1406KB)( 61 )

Fig. & Tab. | References | Supporting Info. | Related Articles | Metrics

Efficient Hydrogenation of Ketones to Alcohols Catalysed by Phosphinoamine Rhenium Complexes

Fang Xiaolong, Wang Jun, Xu Shuting, Li Hao, Hu Kun, Chen, Yiyu

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 241-249 DOI: 10.6023/cjoc202506024

Abstract( 77) HTML( 0) PDF(1153KB)( 18 )

Fig. & Tab. | References | Supporting Info. | Related Articles | Metrics

Design, Synthesis and Anticancer Activity Evaluation of Novel Nitrogen-Containing Heterocyclic Compounds Based on Nitidine Skeleton

Su Xiaowei, Xu Hao, Zhou Huafeng, Wang Xiajie, Li Peiyuan, Xia Xing, Chen Wenya, Huo Lini

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 250-265 DOI: 10.6023/cjoc202504032

Abstract( 58) HTML( 0) PDF(8842KB)( 19 )

Fig. & Tab. | References | Supporting Info. | Related Articles | Metrics

Nickel/Visible Light Dual-Catalyzed C—O Bond Coupling Reactions of Aryl Bromides with Alcohols

Gao Shan, Xie Xin, Liu Yuanhong

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 266-278 DOI: 10.6023/cjoc202506009

Abstract( 54) HTML( 0) PDF(731KB)( 32 )

Fig. & Tab. | References | Supporting Info. | Related Articles | Metrics

Synthesis of α,β-Disubstituted Acrylates via PPh₃-Catalyzed Ring-Opening Addition Reaction of Cyclopropenones with Alkyl Bromides at Room Temperature

Xu Cheng, Peng Tao, Zhou Mengyuan, Liu Minglin, Huang Xiaoqing, Wang Yongfeng, Liu Zheng, Yin Guodong

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 279-288 DOI: 10.6023/cjoc202505033

Abstract( 91) HTML( 0) PDF(733KB)( 53 )

Fig. & Tab. | References | Supporting Info. | Related Articles | Metrics

Characterization of Glutarimide Derivatives from Agrimonia pilosa-Associated Endophytic Streptomyces sp. YINM00048

Su Yuying, Wang Yingfang, Yi Mengzhuo, Zhao Lixing, Li Jiaxuan, Ma Ling, Yin Min

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 289-294 DOI: 10.6023/cjoc202506015

Abstract( 83) HTML( 0) PDF(1592KB)( 35 )

Fig. & Tab. | References | Supporting Info. | Related Articles | Metrics

Activation of the Biosynthetic Gene Cluster in Streptomyces sp. YINM00050 Facilitated the Discovery of a Novel Benzoisochromanequinone

Zhang Yuan, Guo Ying, Yang Mingxi, Dong Kui, Zhao Lixing, Ma Ling, Yin Min

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 295-299 DOI: 10.6023/cjoc202506021

Abstract( 63) HTML( 0) PDF(1166KB)( 13 )

Fig. & Tab. | References | Supporting Info. | Related Articles | Metrics

Two New Linear Furocoumarins from Notopterygium incisum and Their Anti-inflammatory Activity

Hu Su, Zhao Lilian, Li Xinyu, Ye Yubei, Deng Yun, Huang Lijun, Guo Dale

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 300-303 DOI: 10.6023/cjoc202505002

Abstract( 67) HTML( 0) PDF(411KB)( 20 )

Fig. & Tab. | References | Supporting Info. | Related Articles | Metrics

HIGHLIGHTS

Chiral Bicyclic Imidazole-Catalyzed Phosphorus Atom Activation and Asymmetric Construction of Diverse P(V) Compounds

Wu Xiuli, Wu Xingxing

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 304-305 DOI: 10.6023/cjoc202600001

Abstract( 2) HTML( 0) PDF(425KB)( 2 )

Fig. & Tab. | References | Related Articles | Metrics

Chiral Octahedral Cobalt(III)-Catalyzed C—H Macrocyclization to Access Planar-Chiral Cyclophanes

Wen Yilu, Zhao Changgui

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 306-307 DOI: 10.6023/cjoc202600002

Abstract( 4) HTML( 0) PDF(462KB)( 3 )

Fig. & Tab. | References | Related Articles | Metrics