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Base-Promoted, Metal- and Oxidant-Free C=C Bond Cleavage in Enaminones...
Wang Guodong, Guo Yanhui, Wan Jieping

The C=C double bond cleavage of NH2-functionalized enaminones has been realized at room temperature to provide various N-sulfonyl amidines by reacting with sulfonyl azides. The react...

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Nickel-Catalyzed Negishi Coupling of Cyclobutanone Oxime Esters with A...
Shuai Bin, Li Zhao-Ming, Qiu Hui, Fang Ping, Mei Tian-Sheng

A nickel-catalyzed Negishi coupling of cyclobutanone oxime esters with aryl zinc reagents has been developed, in which nickel serves both as an initiator for imine radicals and a catalyst for the coup...

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Asymmetric Transfer Hydrogenation via Dynamic Kinetic Resolution for t...
Zhang Qiying, Zhang Yiming, Hao Erjun, Bai Juan, Qu Guirong, Guo Haiming

N3-Purine nucleoside can be employed as a potent dual inhibitor to inhibit viruses more effectively because it could be possibly recognized by both purine-and pyrimidine-metabolizing...

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  • 2026, 46(1)

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    • 15 2019-11
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    • Recent Advances on the Functionalization of Azlactones at Different Reactive Sites

      Jiang Zhijie, Chen Jinxiu, Zhu Xiaofei, Deng Xinhao, Yan Qiongjiao, Wang Wei, Zhou Hui

      2026, 46 (1), pp 1-20

      DOI: 10.6023/cjoc202506007

      Abstract HTML PDF
    • Recent Progress in the Total Synthesis of abeo-Steroids

      Zhao Lilin, Li Zhaoqi, Zhong Liping, Min Long

      2026, 46 (1), pp 21-38

      DOI: 10.6023/cjoc202506022

      Abstract HTML PDF
    • Structural Modifications, Structure-Activity Relationships, and Total Synthesis Advances in Erythromycin Analogs against Resistant Pathogens

      Cui Xinyi, Guo Lifan, Ma Congxuan, Li Yun, Liang Jianhua

      2026, 46 (1), pp 39-73

      DOI: 10.6023/cjoc202506020

      Abstract HTML PDF
    • Progress in the Synthesis and Biological Studies of S-1-Propenyl-L-cysteine from Garlic

      Tian Lingyan, Wang Shoufeng, Zeng Wei

      2026, 46 (1), pp 74-86

      DOI: 10.6023/cjoc202505028

      Abstract HTML PDF
    • Synthesis of Thiochromone Formamide Derivatives and Their Antifungal Activities

      Zhou Pu, Su Ziyang, Cui Deyun, Cheng Yi-Nan, Li Yi, Zhou Haifeng, Sun Bingjian, Li Honglian

      2026, 46 (1), pp 87-95

      DOI: 10.6023/cjoc202506027

      Abstract HTML PDF
    • Study on the Cyclopropanation Reactivity and Selectivity of Spiroannulated Pentacyclic Diastereoisomers toward Synthesizing Cryptoquinonemethides

      Zhang Yuanhe, Shen Yunjie, Tan Dongxing, Han Fushe

      2026, 46 (1), pp 96-105

      DOI: 10.6023/cjoc202508010

      Abstract HTML PDF
    • Study on the Synthesis and Fungicidal Activity of 1-Azolyl-1,1- diarylmethanes Containing Pyridine Ring

      Hong Sai, Yin Fahong, Chen Minghui, Fu Bin, Xiao Yumei, Qin Zhaohai

      2026, 46 (1), pp 106-117

      DOI: 10.6023/cjoc202506035

      Abstract HTML PDF
    • Silver-Catalyzed Tandem Decarboxylative Cyclization of 2,2-Difluoro-2-(phenylthio)acetic Acids with 2-Aryl-N-acrylamide Indoles

      Liu Jiale, Tang Yucai, Yin Qiumei, Huang Jiaming, Deng Shiqiang, Xia Weiming, Jiang Jie, Wang Zu-Li

      2026, 46 (1), pp 118-127

      DOI: 10.6023/cjoc202507011

      Abstract HTML PDF
    • Synthesis and Characterization of Silacyclopropenes

      Chen Yilin, Yue Jiayi, Lin Yiming, Liu Bingni, Dai Wen, Zhu Hongping

      2026, 46 (1), pp 128-134

      DOI: 10.6023/cjoc202506023

      Abstract HTML PDF
    • Visible-Light-Driven Halogen-Bond-Induced Direct Coupling of Diethyl α-Iodomethylphosphonates with Coumarins/Quinolinones

      Liang Jiarui, Li Jinlan, Jiang Yun, Yao Qiuli, Xu Yingshu, Wang Anjun

      2026, 46 (1), pp 135-145

      DOI: 10.6023/cjoc202506016

      Abstract HTML PDF
    • Regio-reversed [3+2] Cycloaddition of Triketone Enones with Nitrones

      Han Tianjiao, Shi Qianqian, Fu Yundong, Mei Guangjian

      2026, 46 (1), pp 146-155

      DOI: 10.6023/cjoc202507022

      Abstract HTML PDF
    • Heterogeneous Copper Catalyzed Aerobic Oxidative Cross-Coupling of Tertiary Amines with Alkynes

      Tan Ziyun, Yang Xin, Gong Shaofeng, Yang Huiling, Xie Yongyan, Zhang Jingya, Feng Zhetai, Li Wenyi, Xiao Xinsheng

      2026, 46 (1), pp 156-166

      DOI: 10.6023/cjoc202504020

      Abstract HTML PDF
    • Copper-Catalyzed Asymmetric Oxidative Homocoupling Reaction of 3-Hydroxy-2-naphthoates: Design and Optimization of Amino Acid-Based Ligands

      Wang Wen-Long, Wen Jia-Xu, Chen Fei, Bo Chunbo, Li Min, Liu Ning, Du Zhi-Hong

      2026, 46 (1), pp 167-180

      DOI: 10.6023/cjoc202505013

      Abstract HTML PDF
    • Four-Component Hydroxythiolation of Styrenes with Imidazopyridines and Potassium Thiocyanate

      Wang Yu, Huang Hongkun, Ling Chun, Chen Tian, Yao Hua, Yan Zhaohua

      2026, 46 (1), pp 181-188

      DOI: 10.6023/cjoc202506001

      Abstract HTML PDF
    • S-Heteroarylation of Cysteines

      Zhang Xin, Li Fei, Zhou Chenxing, Huo Congde

      2026, 46 (1), pp 189-198

      DOI: 10.6023/cjoc202506011

      Abstract HTML PDF
    • Study on FeCl3-Mediated Reaction of Aryl Boronic Esters with Electrophiles

      Cui Lihua, Li Yatong, Wang Qifeng

      2026, 46 (1), pp 199-206

      DOI: 10.6023/cjoc202506018

      Abstract HTML PDF
    • Nickel-Catalyzed Borylation of Aryl Nonaflates for the Efficient Synthesis of Arylboronates via C—O Bond Functionalization

      Liang Yuan, Gui Chao, Wang Wenwen, Chu Xueqiang, Xu Hao, Shen Zhiliang

      2026, 46 (1), pp 207-214

      DOI: 10.6023/cjoc202507010

      Abstract HTML PDF
    • Photocatalytic Radical-Mediated Synthesis of Unnatural α-Amino Acids from Heteroaryl Aldehydes

      Ren Ke, Zhang Guanglu, Niu Yifan, Wang Xiaomeng, Chen Canyu, Jiang Min

      2026, 46 (1), pp 215-224

      DOI: 10.6023/cjoc202507030

      Abstract HTML PDF
    • PPh3-Mediated One-Pot Synthesis of Indolin-3-ones from 2-Alkynylnitrobenzenes and Indoles

      Feng Faxiu, Xu Shijie, Wang Xue, Yang Zhuoran, Wang Wenjun, Huang Shenlin, Zhang Xiaoxiang

      2026, 46 (1), pp 225-232

      DOI: 10.6023/cjoc202506013

      Abstract HTML PDF
    • Schiff Base Type Fe(III) Complexes Catalyzed Carbon Dioxide and Epoxides for Preparing Cyclic Carbonates

      Liu Tao, Zhou Yongbo, Lang Tongqing, Niu Haibo, Chen Fei, Du Zhihong, Bo Chunbo, Li Min, Liu Ning

      2026, 46 (1), pp 233-240

      DOI: 10.6023/cjoc202506003

      Abstract HTML PDF
    • Efficient Hydrogenation of Ketones to Alcohols Catalysed by Phosphinoamine Rhenium Complexes

      Fang Xiaolong, Wang Jun, Xu Shuting, Li Hao, Hu Kun, Chen, Yiyu

      2026, 46 (1), pp 241-249

      DOI: 10.6023/cjoc202506024

      Abstract HTML PDF
    • Design, Synthesis and Anticancer Activity Evaluation of Novel Nitrogen-Containing Heterocyclic Compounds Based on Nitidine Skeleton

      Su Xiaowei, Xu Hao, Zhou Huafeng, Wang Xiajie, Li Peiyuan, Xia Xing, Chen Wenya, Huo Lini

      2026, 46 (1), pp 250-265

      DOI: 10.6023/cjoc202504032

      Abstract HTML PDF
    • Nickel/Visible Light Dual-Catalyzed C—O Bond Coupling Reactions of Aryl Bromides with Alcohols

      Gao Shan, Xie Xin, Liu Yuanhong

      2026, 46 (1), pp 266-278

      DOI: 10.6023/cjoc202506009

      Abstract HTML PDF
    • Synthesis of α,β-Disubstituted Acrylates via PPh3-Catalyzed Ring-Opening Addition Reaction of Cyclopropenones with Alkyl Bromides at Room Temperature

      Xu Cheng, Peng Tao, Zhou Mengyuan, Liu Minglin, Huang Xiaoqing, Wang Yongfeng, Liu Zheng, Yin Guodong

      2026, 46 (1), pp 279-288

      DOI: 10.6023/cjoc202505033

      Abstract HTML PDF
    • Characterization of Glutarimide Derivatives from Agrimonia pilosa-Associated Endophytic Streptomyces sp. YINM00048

      Su Yuying, Wang Yingfang, Yi Mengzhuo, Zhao Lixing, Li Jiaxuan, Ma Ling, Yin Min

      2026, 46 (1), pp 289-294

      DOI: 10.6023/cjoc202506015

      Abstract HTML PDF
    • Activation of the Biosynthetic Gene Cluster in Streptomyces sp. YINM00050 Facilitated the Discovery of a Novel Benzoisochromanequinone

      Zhang Yuan, Guo Ying, Yang Mingxi, Dong Kui, Zhao Lixing, Ma Ling, Yin Min

      2026, 46 (1), pp 295-299

      DOI: 10.6023/cjoc202506021

      Abstract HTML PDF
    • Two New Linear Furocoumarins from Notopterygium incisum and Their Anti-inflammatory Activity

      Hu Su, Zhao Lilian, Li Xinyu, Ye Yubei, Deng Yun, Huang Lijun, Guo Dale

      2026, 46 (1), pp 300-303

      DOI: 10.6023/cjoc202505002

      Abstract HTML PDF
    • Chiral Bicyclic Imidazole-Catalyzed Phosphorus Atom Activation and Asymmetric Construction of Diverse P(V) Compounds

      Wu Xiuli, Wu Xingxing

      2026, 46 (1), pp 304-305

      DOI: 10.6023/cjoc202600001

      Abstract HTML PDF
    • Chiral Octahedral Cobalt(III)-Catalyzed C—H Macrocyclization to Access Planar-Chiral Cyclophanes

      Wen Yilu, Zhao Changgui

      2026, 46 (1), pp 306-307

      DOI: 10.6023/cjoc202600002

      Abstract HTML PDF
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ISSN: 0253-2786 CN: 31-1321/06

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