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Chinese Journal of Organic Chemistry >

2013 , Vol. 33 >Issue 01: 101 - 105

DOI: https://doi.org/10.6023/cjoc201208019

Articles

Synthesis and Fungicidal Activity of 1,3,4-Oxadiazole Derivatives Containing Pyrazole Moiety

  • Sun Nabo ,
  • Tong Jianying ,
  • Wu Hongke
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  • a College of Biology and Environmental Engineering, Zhejiang Shuren University, Hangzhou 310015;
    b College of Chemical Engineering and Materials Science, Zhejiang University of Technology, Hangzhou 310014

Received date: 2012-08-20

  Revised date: 2012-10-07

  Online published: 2012-10-12

Supported by

Project supported by the Program of Education Department of Zhejiang Province (No. Y200803060).

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Abstract

A series of novel 1,3,4-oxadiazole derivatives were synthesized from acetylacetone, hydrazine hydrate by multi-step reactions. Their structures were characterized by 1H NMR, MS and elemental analyses. The target compounds were evaluated for their fungicidal activities against Corynespora cassiicola, Pseudomonas syringae pv. Lachrymans, Pseudoperonospora cubensis and Sclerotinia sclerotiorum in vivo, and the results indicated that some of the title compounds displayed excellent fungicidal activities.

Key words： 1,3,4-oxadiazole; pyrazole; synthesis; fungicidal activity

Cite this article

Sun Nabo , Tong Jianying , Wu Hongke . Synthesis and Fungicidal Activity of 1,3,4-Oxadiazole Derivatives Containing Pyrazole Moiety[J]. Chinese Journal of Organic Chemistry, 2013 , 33(01) : 101 -105 . DOI: 10.6023/cjoc201208019

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