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Chinese Journal of Organic Chemistry >

2013 , Vol. 33 >Issue 11: 2396 - 2401

DOI: https://doi.org/10.6023/cjoc201305024

Articles

Synthesis and Herbicidal Activities of 1-Methylcyclohexyl-formayl Thioureas

  • Gong Yunyun ,
  • Huang Wei ,
  • Liu Xinghai ,
  • Weng Jianquan ,
  • Tan Chengxia
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  • College of Chemical Engineering and Materials Science, Zhejiang University of Technology, Hangzhou 310014

Received date: 2013-05-14

  Revised date: 2013-06-27

  Online published: 2013-07-10

Supported by

Project supported by the The Twelfth Five-Year National Key Technology R & D Project (No. 2011BAE06B03-01).

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Abstract

In order to find out novel pesticide lead compounds with good biological activity, totally 24 novel 1-methylcyclo-hexyl-formyl thiourea compounds were synthesized by the reaction of 1-methylcyclohexane-carbonyl chloride with various substituted amines. Their structures were confirmed by 1H NMR, MS, and elemental analysis. The biological activities of these compounds were evaluated. Most of the compounds showed good herbicide activities at the concentration of 200 mg/L.

Key words： 1-methylcyclohexyl; acyl thiourea; synthesis; herbicidal activity

Cite this article

Gong Yunyun , Huang Wei , Liu Xinghai , Weng Jianquan , Tan Chengxia . Synthesis and Herbicidal Activities of 1-Methylcyclohexyl-formayl Thioureas[J]. Chinese Journal of Organic Chemistry, 2013 , 33(11) : 2396 -2401 . DOI: 10.6023/cjoc201305024

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