Studies on acyl thiosemicarbazides and related heterocyclic compounds VI: Syntheses of 3-(4'-pyridinyl)-4-aryl-1,2,4-triazol-5-yl sulphides

Chin. J. Org. Chem. ›› 1988, Vol. 8 ›› Issue (2): 131-133. Previous Articles Next Articles

酰胺基硫脲及其相关杂环化合物的研究 VI:3-(4'-吡啶基)-4-芳基-1,2,4-三唑-5-烃硫醚类化合物的合成

张自义;杨珂新

兰州大学化学系

发布日期:1988-04-25

Studies on acyl thiosemicarbazides and related heterocyclic compounds VI: Syntheses of 3-(4'-pyridinyl)-4-aryl-1,2,4-triazol-5-yl sulphides

ZHANG ZIYI;YANG KEXIN

Published:1988-04-25

Abstract

Title compounds I (R = substituted Ph, a-naphthyl, R1 = Me, CH2CO2Et) were prepared in 54-90% yield by treating triazolinethiones II with MeI or ClCH2CO2Et in alkaline media.

Key words: PYRIDINE P, THIOKETONE, AMIDES, ANTICARCINOGEN, SUBSTITUTION REACTION, THIOUREAS, SULFUR ETHER, NUCLEOPHILIC REACTION, TAUTOMERISM, PYRRODIAZOLE P

CLC Number:

O621

Cite this article

ZHANG ZIYI;YANG KEXIN. Studies on acyl thiosemicarbazides and related heterocyclic compounds VI: Syntheses of 3-(4'-pyridinyl)-4-aryl-1,2,4-triazol-5-yl sulphides[J]. Chin. J. Org. Chem., 1988, 8(2): 131-133.

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酰胺基硫脲及其相关杂环化合物的研究 VI:3-(4'-吡啶基)-4-芳基-1,2,4-三唑-5-烃硫醚类化合物的合成

Studies on acyl thiosemicarbazides and related heterocyclic compounds VI: Syntheses of 3-(4'-pyridinyl)-4-aryl-1,2,4-triazol-5-yl sulphides

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