A new convienent synthesis of  3-substituted-(1H)-pyrimidine [1, 2-a] quinoline-1-ones and  2-substituted pyrimidine [1, 2-a] benzoimidazole-4-(10H)-ones

Chin. J. Org. Chem. ›› 1993, Vol. 13 ›› Issue (5): 518-522. Previous Articles Next Articles

Original Articles

3-取代-(1H)-嘧啶[1, 2-a]喹啉-1-酮和2-取代嘧啶[1, 2a]苯骈咪唑-4-(10H)- 酮的简便合成法

黄宪;叶芳尘

杭州大学化学系.杭州(310028);温州师范学院化学系.温州(325003)

发布日期:1993-10-25

A new convienent synthesis of 3-substituted-(1H)-pyrimidine [1, 2-a] quinoline-1-ones and 2-substituted pyrimidine [1, 2-a] benzoimidazole-4-(10H)-ones

Huang Xian;Ye Fangchen

Hangzhou Univ., Dept of Chem.Hangzhou(310028);Wenzhou Normal Coll, Dept Chem.Wenzhou(325003)

Published:1993-10-25

Abstract

2-Aminoquinoline reacted with 5-bismethylthiomethylene or 5- methylthioalkylidene isopropylidene malonates as one pot reaction to afford a new convienent systhesis of 3-substituted-(1H)-pyrimdine [1, 2-a] quinoline-1-ones. 2-Aminobenzoimidazole could also take place analogous reaction to give 2-substituted pyrimidine [1, 2-a] benzoimidazole-4-(10H)-ones.

Key words: QUINOLINE, AMINOQUINOXALINE, PYRIMIDONE, NUCLEOPHILIC REAGENTS, SYNTHESIS METHODS

CLC Number:

O621

Cite this article

Huang Xian;Ye Fangchen. A new convienent synthesis of 3-substituted-(1H)-pyrimidine [1, 2-a] quinoline-1-ones and 2-substituted pyrimidine [1, 2-a] benzoimidazole-4-(10H)-ones[J]. Chin. J. Org. Chem., 1993, 13(5): 518-522.

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3-取代-(1H)-嘧啶[1, 2-a]喹啉-1-酮和2-取代嘧啶[1, 2a]苯骈咪唑-4-(10H)- 酮的简便合成法

A new convienent synthesis of 3-substituted-(1H)-pyrimidine [1, 2-a] quinoline-1-ones and 2-substituted pyrimidine [1, 2-a] benzoimidazole-4-(10H)-ones

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3-取代-(1H)-嘧啶[1, 2-a]喹啉-1-酮和2-取代嘧啶[1, 2a]苯骈 咪唑-4-(10H)- 酮的简便合成法

A new convienent synthesis of 3-substituted-(1H)-pyrimidine [1, 2-a] quinoline-1-ones and 2-substituted pyrimidine [1, 2-a] benzoimidazole-4-(10H)-ones

Knowledge

Abstract

Cite this article

share this article

References

Related Articles 15

Recommended Articles

Metrics

Comments

3-取代-(1H)-嘧啶[1, 2-a]喹啉-1-酮和2-取代嘧啶[1, 2a]苯骈咪唑-4-(10H)- 酮的简便合成法