Chin. J. Org. Chem. ›› 2018, Vol. 38 ›› Issue (4): 775-790.DOI: 10.6023/cjoc201709044 Previous Articles     Next Articles

Special Issue: 碳氢活化合辑2018-2019



金城安a, 徐庆a, 冯高峰a, 金阳a,b, 张连阳b,c   

  1. a 绍兴文理学院化学化工学院 绍兴 312000;
    b 绍兴文理学院 浙江省清洁染整技术研究重点实验室 绍兴 312000;
    c 绍兴文理学院纺织服装学院 绍兴 312000
  • 收稿日期:2017-09-26 修回日期:2017-11-08 发布日期:2017-11-17
  • 通讯作者: 张连阳
  • 基金资助:


Progress in C—H Bond Functionalization on C-3 Position of Imidazo[1,2-a] pyridines

Jin Cheng'ana, Xu Qinga, Feng Gaofenga, Jin Yanga,b, Zhang Lianyangb,c   

  1. a College of Chemistry and Chemical Engineering, Shaoxing University, Shaoxing 312000;
    b Key Laboratory of Clean Dyeing and Finishing Technology of Zhejiang Province, Shaoxing University, Shaoxing 312000;
    c College of Textile and Garment, Shaoxing University, Shaoxing 312000
  • Received:2017-09-26 Revised:2017-11-08 Published:2017-11-17
  • Contact: 10.6023/cjoc201709044
  • Supported by:

    Project supported by the Research Project of Shaoxing University (No. 2016LG1011).

3-Substituted imidazo[1,2-a] pyridines are important N-fused heterocycles with extensive application value in medicine, materials and other fields. C(3)-H bond functionalization strategy was a simple and effective way to build 3-substituted imidazo[1,2-a] pyridines. The recent advances of the access to 3-substituted imidazo[1,2-a] pyridines according to the type of bonding (C-C, C-S/Se, C-N/P) on C-3 position are briefly summarized, and a prospect for the future development is made.

Key words: 3-substituted imidazo[1,2-a] pyridine, C-H bond functionalization, C-3 position