铑催化碳氢二氟烯丙基化/
N-碘代丁二酰亚胺介导的环化反应构建含氟3,4-二氢嘧啶并[1,6-
a]吲哚-1(2
H)-酮衍生物
赵森, 李淳朴, 许斌, 柳红
Cp*Rh(III)-Catalyzed C—H 3,3-Difluoroallylation of Indoles and
N-Iodosuccinimide-Mediated Cyclization for the Synthesis of Fluorinated 3,4-Dihydropyrimido-[1,6-
a]-indol-1(2
H)-one Derivatives
Zhao Sen, Li Chunpu, Xu Bin, Liu Hong
有机化学
.
2020, (6): 1549
-1562
.
DOI: 10.6023/cjoc202004039