基于ABBV-075的新型溴结构域蛋白4 (BRD4)小分子抑制剂的设计、合成及活性评价
徐晨淏, 龚云鹏, 陈雅欣, 宋启梦, 李娇, 郑一超, 李雯, 孙凯, 刘宏民
Design, Synthesis and Activity Evaluation of Novel Bromodomain-Containing Protein 4 (BRD4) Small Molecule Inhibitor Based on ABBV-075
Chenhao Xu, Yunpeng Gong, Yaxin Chen, Qimeng Song, Jiao Li, Yichao Zheng, Wen Li, Kai Sun, Hongmin Liu
有机化学 . 2021, (4): 1712 -1721 .  DOI: 10.6023/cjoc202007059