Chin. J. Org. Chem. ›› 2018, Vol. 38 ›› Issue (2): 504-508.DOI: 10.6023/cjoc201708054 Previous Articles     Next Articles



王彬a, 叶文波a, 晏子聪b, 万常峰a, 侯豪情a, 汪志勇b   

  1. a 江西师范大学化学化工学院 南昌 330022;
    b 中国科学技术大学化学系 合肥 230026
  • 收稿日期:2017-08-25 修回日期:2017-10-11 发布日期:2017-10-24
  • 通讯作者: 万常峰
  • 基金资助:


A New Catalyst-Free Synthesis of 2,3-Dicarboxylic Ester Quinoline Derivatives

Wang Bina, Ye Wenboa, Yan Zicongb, Wan Changfenga, Hou Haoqinga, Wang Zhiyongb   

  1. a College of Chemistry and Chemical Engineering, Jiangxi Normal University, Nanchang 330022;
    b Department of Chemistry, University of Science and Technology of China, Hefei 230026
  • Received:2017-08-25 Revised:2017-10-11 Published:2017-10-24
  • Contact: 10.6023/cjoc201708054
  • Supported by:

    Project supported by the National Natural Science Foundation of China (Nos. 21402068, 21574060, 21472177).

A high efficient method for the synthesis of 2, 3-dicarboxylic ester quinoline derivatives which employed o-amino diphenyl methylone derivatives and acetylenedicarboxylic esters as the reaction substrates was developed. This method possessed the character of catalyst-free and mild reaction conditions. Proposed mechanism was also studied according to the reaction result.

Key words: quinoline derivatives, catalyst-free, green synthesis