Synthesis of  N'-4,5,6trisubstituted-2-pyrimidin-yl-N-2- sulfonylbenzoyl-imino  acetylureas

Abstract

Eleven new compounds were designed and synthesined using "Substrmture Link Wory" according to the bioisosterism principles. Their structures were confirmed by IR、^1H NMR、 MS and elemental analysis. The preliminary results of biological activity test showed that some of them had good biological activities against root of rape.

Key words: PYRIMIDINE P, PHENYL UREA GROUP HERBICIDES, TRIHEXYPHENIDYL, BENZENESULFONAMIDE P, PLANT GROWTH REGULATORS, BIOLOGICAL ACTIVITY, SPECTROMETRIC ANALYSIS

CLC Number:

TQ45

Cite this article

Xue Sijia;Wang Tao;Liao Zhanru. Synthesis of N'-4,5,6trisubstituted-2-pyrimidin-yl-N-2- sulfonylbenzoyl-imino acetylureas[J]. Chin. J. Org. Chem., 2000, 20(5): 731-734.

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N'-4,5,6-三取代嘧啶-2-基-N-邻磺酰苯甲酰亚胺基乙酰脲的合成(Ⅰ)