综述与进展

5-氨基噻唑衍生物合成的研究进展

  • 钟世华 ,
  • 杨柱 ,
  • 范明亮 ,
  • 张沐 ,
  • 刘建兵
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  • 湖南师范大学化学化工学院 长沙 410081

收稿日期: 2011-07-04

  修回日期: 2011-11-04

  网络出版日期: 2012-03-09

Progress in the Synthesis of 5-Aminothiazole Derivatives

  • ZHONG Shi-Hua ,
  • YANG Zhu ,
  • FAN Ming-Liang ,
  • ZHANG Mu ,
  • LIU Jian-Bing
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  • College of Chemistry and Chemical Engineering, Hunan Normal University, Changsha 410086

Received date: 2011-07-04

  Revised date: 2011-11-04

  Online published: 2012-03-09

摘要

5-氨基噻唑衍生物具有很好的生理活性, 其合成方法和生物生理活性研究已引起药物研发者的关注. 综述了近几十年来有关5-氨基噻唑衍生物的合成方法.

本文引用格式

钟世华 , 杨柱 , 范明亮 , 张沐 , 刘建兵 . 5-氨基噻唑衍生物合成的研究进展[J]. 有机化学, 2012 , 32(02) : 230 -238 . DOI: 10.6023/cjoc1107041

Abstract

5-Aminothiazole derivatives possess good physiological activities. Their synthesis and study of bioactivities have recently attracted increasingly more attention. In this paper, the synthetic methods of 5-aminothiazole derivatives are reviewed and evaluated.

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