Chin. J. Org. Chem. ›› 2016, Vol. 36 ›› Issue (9): 2024-2038.DOI: 10.6023/cjoc201603034 Previous Articles     Next Articles



李闪闪, 洪海龙, 竺宁, 韩利民, 吕佳媛   

  1. 内蒙古工业大学化工学院 呼和浩特 010051
  • 收稿日期:2016-03-20 修回日期:2016-05-06 发布日期:2016-05-19
  • 通讯作者: 洪海龙, 竺宁;
  • 基金资助:


Review About the Synthesis of 1,3-Benzothiazinone Derivatives

Li Shanshan, Hong Hailong, Zhu Ning, Han Limin, Lü Jiayuan   

  1. Chemical Engineering College, Inner Mongolia University of Technology, Hohhot 010051
  • Received:2016-03-20 Revised:2016-05-06 Published:2016-05-19
  • Supported by:

    Project supported by the National Natural Science Foundation of China (Nos.21362019, 21666026), the Natural Science Foundation of Inner Mongolia (No.2016MS0207) and the Graduate Student Scientific Research Innovation Foundation of the Department of Education of Inner Mongolia Autonomous Region (No.S20151012805).

1,3-Benzothiazinone derivatives have widely bioactivities. So the methods for the synthesis of these 1,3-benzothiazinone derivatives have attracted enormous attentions worldwide. From the method of introducing sulfur atom and the reaction mechanism for the formation of benzothiazinone derivatives, the method of synthesizing 1,3-benzothiazinone derivatives has been summarized in this review. So the thiophenol derivatives, disulfide derivatives, the same carbon connected with amino and mercapto derivatives, isothiocyanate derivatives and some smaller sulfur molecules are used as starting materials.

Key words: 1,3-benzothiazinone, sulfur source, synthetic methods, reaction mechanism