有机化学 ›› 1999, Vol. 19 ›› Issue (4): 390-394. 上一篇    下一篇

研究论文

1-取代酰基-4-磷酰基氨基硫脲及其1, 3, 4-恶二唑杂环衍生物 的合成

卢水明;陈茹玉   

  1. 南开大学元素有机化学研究所.天津(300071)
  • 发布日期:1999-08-25

The synthesis of 1-acyl-4-phosphoryl thiosemicarbazides and their heterocyclic derivatives of 1, 3, 4-oxadiazoles

Lu Shuiming;Chen Ruyu   

  1. Nankai Univ, Elementoorgan Chem Lab.Tianjin(300071)
  • Published:1999-08-25

合成了1-取代酰基-4-磷酰基氨基硫脲(5),以及由(5)衍生的环化产物2-磷酰氨基-5-苯基(或氰乙基)-1,3,4-恶二唑(6),它们的结构经^1HNMR,IR和元素分析的证实。初步生测结果表明,部分化事物具有一定的植物生长调节活性和除草活性。

关键词: 植物生长调节活性, 合成, 生物活性, 除草活性, 恶二唑, 氨基硫脲, 磷酰基

1-Acyl-4-phosphoryl thiosemicarbazides (5) and their heterocyclic derivatives of 1, 3, 4-oxadiazoles (6) were synthesized, whose structures were confirmed by ^1H NMR, IR and elemental analysis. The general screening results showed that some of them had plant growth regulator and herbicidal activity.

Key words: FURODIAZOLE (=OXDIAZOLE), SYNTHESIS, THIOSEMICARBAZIDE, BIOLOGICAL ACTIVITY, PHOSPHORYL

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