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有机化学
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有机化学 ›› 2008, Vol. 28 ›› Issue (01): 17-28. 上一篇    下一篇

综述与进展

α-氰基丙烯酸酯及其衍生物的合成与农药生物活性研究进展

张慧苹，宋宝安*，王献友，龙宁，胡德禹，杨松
薛伟，卢平，金林红   

  1. (贵州大学精细化工研究开发中心 教育部绿色农药与生物工程重点实验室 贵阳 550025)
  • 收稿日期:2006-08-21 修回日期:1900-01-01 发布日期:2008-01-23
  • 通讯作者: 宋宝安

Recent Advances in the Synthesis and Biological Activity on Pesticide of α-Cyanoacrylates and Its Analognes

ZHANG Hui-Ping, SONG Bao-An*, WANG Xian-You, LONG Ning
HU De-Yu, YANG Song, XUE Wei, LU Ping, JIN Lin-Hong   

  1. (Key Laboratory of Green Pesticide and Bioengineering, Ministry of Education, Center for Research and Development of Fine Chemicals, Guizhou University, Guiyang 550025)
  • Received:2006-08-21 Revised:1900-01-01 Published:2008-01-23
  • Contact: SONG Bao-An

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丙烯酸酯是一类具有良好生物活性的化合物, 由于它作用机制新颖、环境友好, 故其分子设计和合成及生物活性成为目前农药创制的热点之一, 按其在农药应用方面的不同活性作用进行分类, 综述了丙烯酸酯及其类似物的合成、生物活性与除草活性方面构效关系的研究进展.

关键词: 丙烯酸酯, 合成, 生物活性, 构效关系

Cyanoacrylates and their analogues are an important class of compounds with high bioactivities. Recently, studies on the molecular designing, synthesizing and bioactivities of α-cyanoacrylates have attracted more and more attentions according to their characteristics of novel mechanism and friendly-environment. Recent advances in the synthesis, structure, biological activity and structure-activity relationships (SAR) of 2-cyanoacrylate and its analogues are reviewed emphatically on their applying on pesticide based on different bioactivities.

Key words: synthesis, acrylate, bioactivity, structure-activity relationships