Synthesis of styryl-substituted hetero-fused troponoid compounds

Abstract

3-(3,4,5-trimethoxy) cinnamoyltropolone and 3-(3,4- methylenedioxy) cinnamoyltropolone reacts with hydroxylamine and phenyldrazine to afford 3-(3,4,5- trimethoxy) styryl-8H-cyclohept [d] isoxazol-8-one, 1-phenyl-3-(3,4-methylenedioxy) styryl-8H-cyclohept [d] isoxazol-8-one, 3-(3,4,5-trimethoxy) styryl-1,8- dihydrocycloheptapyrazol-8-one and 1-phenyl-3-(3,4- methylenedioxy) styryl-1,8-dihydrocycloheptapyrazol-8-one, respectively.

Key words: SYNTHESIS, HETEROCYCLIC COMPOUNDS, ANTITUMOR DRUGS, CONDENSATION

CLC Number:

O621

Cite this article

GAO WENTAO;ZHANG BAOTIAN;SUN SHUGUANG. Synthesis of styryl-substituted hetero-fused troponoid compounds[J]. Chin. J. Org. Chem., 1995, 15(1): 104-106.

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