Chin. J. Org. Chem. ›› 2018, Vol. 38 ›› Issue (4): 738-751.DOI: 10.6023/cjoc201709045 Previous Articles     Next Articles

Special Issue: 元素有机化学合辑2018-2019



徐玉良a,b, 方浩a,b   

  1. a 山东大学 天然产物化学生物学教育部重点实验室 济南 250012;
    b 山东大学药学院 药物化学研究所 济南 250012
  • 收稿日期:2017-09-28 修回日期:2017-11-11 发布日期:2017-12-05
  • 通讯作者: 方浩
  • 基金资助:


Research Progress towards Synthesis of Aryl Boronic Acid Compounds

Xu Yulianga,b, Fang Haoa,b   

  1. Ministry of Education), Shandong University, Jinan 250012;
    b Department of Medicinal Chemistry, School of Pharmacy, Shandong University, Jinan 250012
  • Received:2017-09-28 Revised:2017-11-11 Published:2017-12-05
  • Contact: 10.6023/cjoc201709045
  • Supported by:

    Project supported by the National Natural Science Foundation of China (No. 21672127).

Aromatic boronic acids and esters are essential intermediates and have been widely used in biology, medicine and material science. In this paper, the resent progress on their synthesis is summarized, especially Pd-catalyzed borylation of aryl chlorides with steric hindrance substrates, other metal (Ni, Cu, Fe, Zn, Rh, Co)-catalyzed borylation, metal-free borylation, and photoinduced borylation.

Key words: aromatic boronic acids, metal-catalyzed, metal-free catalyzed, photoinduced