Synthesis and Bioactivity of N′-tert-Butyl-N-substituted Acyl(thio)urea  Derivatives

Chinese Journal of Organic Chemistry ›› 2004, Vol. 24 ›› Issue (2): 227-230. Previous Articles Next Articles

N′-叔丁基-N-取代酰基(硫)脲类化合物的合成及生物活性测定

薛思佳, 柯少勇^*, 段李平

上海师范大学生命与环境科学学院上海 200234

收稿日期:2003-05-26 修回日期:2003-07-07 接受日期:2003-09-01 发布日期:2022-09-20
基金资助:
上海市科委2001科学发展基金(No. BL200116)资助项目

Synthesis and Bioactivity of N′-tert-Butyl-N-substituted Acyl(thio)urea Derivatives

XUE, Si-Jia, KE, Shao-Yong^*, DUAN, Li-Ping

College of Life and Environment Science, Shanghai Normal University, Shanghai 200234

Received:2003-05-26 Revised:2003-07-07 Accepted:2003-09-01 Published:2022-09-20
Contact: * E-mail: keshaoyong@163.com

Abstract

Eight new N′-tert-butyl-N-substituted acylurea and N′-tert-butylaminocarbonyl-N-substituted acylthiourea derivatives were synthesized and characterized. The structures of these compoundswere determined by ¹H NMR, IR and elemental analysis. The preliminary biologic tests show that some of the title compounds have excellent inhibitory activity against weeds.

Key words: N′-tert-butyl-N-substituted acylurea, N′-tert-butylaminocarbonyl-N-substituted acylthiourea, synthesis, biological activity

Cite this article

XUE, Si-Jia, KE, Shao-Yong, DUAN, Li-Ping. Synthesis and Bioactivity of N′-tert-Butyl-N-substituted Acyl(thio)urea Derivatives[J]. Chinese Journal of Organic Chemistry, 2004, 24(2): 227-230.

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N′-叔丁基-N-取代酰基(硫)脲类化合物的合成及生物活性测定

Synthesis and Bioactivity of N′-tert-Butyl-N-substituted Acyl(thio)urea Derivatives

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