Three Component One-Pot Synthesis of Methyl 3-(2-Quinolyl)azulene-1-carboxylates

Chin. J. Org. Chem. ›› 2009, Vol. 29 ›› Issue (06): 979-984. Previous Articles Next Articles

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三组分一锅法合成3-(2-喹啉基)薁甲酸甲酯衍生物

孙曙光 ; 谷峥; 王道林* ; 韩珊黄孝东

(渤海大学化学化工学院辽宁省应用化学重点实验室锦州 121003)

收稿日期:2008-07-14 修回日期:2008-10-23 发布日期:2009-06-20
通讯作者: 王道林

Three Component One-Pot Synthesis of Methyl 3-(2-Quinolyl)azulene-1-carboxylates

Sun, Shuguang ; Gu, Zheng ; Wang, Daolin* ; Han, Shan ; Huang, Xiaodong

(Liaoning Key Laboratory of Applied Chemistry, College of Chemistry and Chemical Engineering,
Bohai University, Jinzhou 121003)

Received:2008-07-14 Revised:2008-10-23 Published:2009-06-20
Contact: Wang, Daolin

Abstract

Methyl 3-(2-quinolyl)azulene-1-carboxylate derivatives were synthesized by three component one-pot condensation of methyl 1-formoylazulene-3-carboxylate, aromatic amines and alkylaldehydes under mild conditions. This method provides several advantages such as good yield and simple work-up procedure. All the products were fully characterized by 1H NMR, IR spectra and elemental analysis.

Key words: 1-formoylazulene-3-carboxylate, 3-(2-quinolyl)azulene, synthesi, azulene

Cite this article

Sun, Shuguang ; Gu, Zheng ; Wang, Daolin* ; Han, Shan ; Huang, Xiaodong. Three Component One-Pot Synthesis of Methyl 3-(2-Quinolyl)azulene-1-carboxylates[J]. Chin. J. Org. Chem., 2009, 29(06): 979-984.

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三组分一锅法合成3-(2-喹啉基)薁甲酸甲酯衍生物

Three Component One-Pot Synthesis of Methyl 3-(2-Quinolyl)azulene-1-carboxylates

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