Synthesis and Herbicidal Activity of Some New Diacylhydrazines De-rivatives Fluoride-Containing Pyrazolyl Moiety

Chin. J. Org. Chem. ›› 2011, Vol. 31 ›› Issue (08): 1295-1299. Previous Articles Next Articles

Notes

含氟代吡唑环的双酰肼类化合物的合成及除草活性

张向阳，李永曙，翁建全，谭成侠*

(浙江工业大学化学工程与材料学院杭州 310014)

收稿日期:2010-09-01 修回日期:2011-02-21 发布日期:2011-03-28
通讯作者: 谭成侠 E-mail:nkulxh@gmail.com

Synthesis and Herbicidal Activity of Some New Diacylhydrazines De-rivatives Fluoride-Containing Pyrazolyl Moiety

ZHANG Xiang-Yang, LI Yong-Shu, WENG Jian-Quan, TAN Cheng-Xia

(College of Chemical Engineering and Materials Science, Zhejiang University of Technology, Hangzhou 310014)

Received:2010-09-01 Revised:2011-02-21 Published:2011-03-28

In search of novel bioactive compounds, compounds 3a～3s were designed and synthesized by introducing the fluoropyrazolyl pharmacophore into the diacylhydrazine scaffold. Their structures were confirmed by ¹H NMR, FTIR, MS techniques and elemental analysis. The herbicidal activities of these compounds were evaluated. The bioassay results showed that most of them exhibited higher herbicidal activities against dicotyledonous weeds (Abutilon theophrasti, Amaranthus ascedense and Amaranthus retroflexus) than monocotyledonous weeds.

Key words: fluoride pyrazole, diacylhydrazine, synthesis, herbicidal activity

Cite this article

ZHANG Xiang-Yang, LI Yong-Shu, WENG Jian-Quan, TAN Cheng-Xia. Synthesis and Herbicidal Activity of Some New Diacylhydrazines De-rivatives Fluoride-Containing Pyrazolyl Moiety[J]. Chin. J. Org. Chem., 2011, 31(08): 1295-1299.

Export EndNote|Reference Manager|ProCite|BibTeX|RefWorks

[1]	Fakai Zou, Nengzhong Wang, Hui Yao, Hui Wang, Mingguo Liu, Nianyu Huang. Regio- and Stereo-selective Synthesis of 1β-/3R-Aryl Thiosugar [J]. Chinese Journal of Organic Chemistry, 2024, 44(2): 593-604.
[2]	Luyao Li, Zhongwen He, Zhenguo Zhang, Zhenhua Jia, Teck-Peng Loh. Application of Triaryl Carbenium in Organic Synthesis [J]. Chinese Journal of Organic Chemistry, 2024, 44(2): 421-437.
[3]	Qinggang Mei, Qinghan Li. Recent Progress of Visible Light-Induced the Synthesis of C(3) (Hetero)arylthio Indole Compounds [J]. Chinese Journal of Organic Chemistry, 2024, 44(2): 398-408.
[4]	Penghui Li, Qingyang Xie, Fuxian Wan, Yuanhong Zhang, Lin Jiang. Synthesis and Fungicidal Activity of Novel Substituted Pyrimidine-5-carboxamides Bearing Cyclopropyl Moiety [J]. Chinese Journal of Organic Chemistry, 2024, 44(2): 650-656.
[5]	Weiqing Yang, Yanbing Ge, Yuanyuan Chen, Ping Liu, Haiyan Fu, Menglin Ma. Design and Synthesis of Fluorescent 1,8-Napthalimide Derivatives and Their Identification of Cysteine [J]. Chinese Journal of Organic Chemistry, 2024, 44(1): 180-194.
[6]	Shihang Yu, Jiawei Liu, Biyu An, Qinghua Bian, Min Wang, Jiangchun Zhong. Asymmetric Synthesis of the Contact Sex Pheromone of Neoclytus acuminatus acuminatus (Fabricius) [J]. Chinese Journal of Organic Chemistry, 2024, 44(1): 301-308.
[7]	Qianfan Zhao, Yongzheng Chen, Shiming Zhang. Application and Mechanism Study of Carbon-Based Metal-Free Catalysts in Organic Synthesis [J]. Chinese Journal of Organic Chemistry, 2024, 44(1): 137-147.
[8]	Shan Chen, Zhilin Chen, Qiong Hu, Yanshuang Meng, Yue Huang, Pingfang Tao, Liru Lu, Guobao Huang. Recognition of Bis-thiourea Tweezers to Neutral Molecules in Non-Polar Solvent [J]. Chinese Journal of Organic Chemistry, 2024, 44(1): 277-281.
[9]	Huakun Wang, Xiaolong Ren, Yining Xuan. Study of the Halide Salt Catalyzed [3＋2] Cycloaddition of α,β-Epoxy Carboxylate with Isocyanate [J]. Chinese Journal of Organic Chemistry, 2024, 44(1): 251-258.
[10]	Yukun Jin, Baoyi Ren, Fushun Liang. Visible Light-Mediated Selective C—F Bond Cleavage of Trifluoromethyl Groups and Its Application in Synthesizing gem-Difluoro-Containing Compounds [J]. Chinese Journal of Organic Chemistry, 2024, 44(1): 85-110.
[11]	Cuiyun Ma, Hailan Luo, Fuhua Zhang, Dan Guo, Shuxing Chen, Fei Wang. Green Biosynthesis, Photophysical Properties and Application of 3-Pyrrolyl BODIPY [J]. Chinese Journal of Organic Chemistry, 2024, 44(1): 216-223.
[12]	Bozhen Wang, Jie Zhang, Chunhui Nian, Mingming Jin, Miaomiao Kong, Wulan Li, Wenfei He, Jianzhang Wu. Synthesis and Antitumor Activity of 3,4-Dichlorophenyl Amides [J]. Chinese Journal of Organic Chemistry, 2024, 44(1): 232-241.
[13]	Ruixia Cao, Yuping Jia. Synthesis and Biological Activity of Novel Pyrrolo[2,3-d]pyrimidine Derivatives Containing Coumarin [J]. Chinese Journal of Organic Chemistry, 2023, 43(9): 3304-3311.
[14]	Huanqing Li, Zhaohua Chen, Zujia Chen, Qiwen Qiu, Youcai Zhang, Sihong Chen, Zhaoyang Wang. Research Progress in Mercury Ion Fluorescence Probes Based on Organic Small Molecules [J]. Chinese Journal of Organic Chemistry, 2023, 43(9): 3067-3077.
[15]	Ran Zhou, Chunmei Yuan, Tao Zhang, Piao Mao, Yi Liu, Kaini Meng, Hui Xin, Wei Xue. Design, Synthesis and Bioactivity of Chalcone Derivative Containing Quinazolinone [J]. Chinese Journal of Organic Chemistry, 2023, 43(9): 3196-3209.

含氟代吡唑环的双酰肼类化合物的合成及除草活性

Synthesis and Herbicidal Activity of Some New Diacylhydrazines De-rivatives Fluoride-Containing Pyrazolyl Moiety

PDF

Knowledge

Cited

Abstract

Cite this article

share this article

References

Related Articles 15

Recommended Articles

Metrics

Comments