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About the Cover:α-Chiral primary amine subunits are widespread structural units in a large number of pharmaceutical molecules and are key intermediates toward the preparation of numerous amine-containing drugs. In this account, systematic studies on direct synthesis of chiral primary amines via met-al-catalyzed asymmetric reductive amination with cheap ammonium salts as amine sources from Xumu Zhang and Qin Yin’s group are summarized on page 2261.
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About the Cover:The recent progress on light-promoted transition metal- catalyzed C-heteroatom coupling reactions is reviewed with emphasis on its development process and reaction mechanism by Song and Xue on page 2275. The current problems and future development prospects in this field are also summarized and prospected.
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