Chinese Journal of Organic Chemistry 2024, 44(11)

- About the Cover:
  
  Selective functionalization of hydrocarbon chains is an important scientific problem in synthetic chemistry, and direct functionaliza-tion of easily available alkanes or alkenes is an ideal method for their efficient and high value-added conversion. A comprehensive overview of the recent developments in se-lective multi-site functionalization of hydro-carbon chains is provided by Wang, Liu, Yang, Wu and Zhang on page 3273.
- About the Cover:
  
  Amidoenol structural fragments are widely found in bioactive natural products and pharmaceutical compounds. The addition reaction of tert-butyl 1-indole- carboxylate and ynamides, catalyzed by Ca(NTf₂)₂, which enables the construction of key indole amidoenol fragments, is reported by Zhang, Song, Li, Zheng and Wei on page 3490. The method demonstrates stable yields, high regioselectivities, and well substrate suitabil-ities.
- About the Cover:
  
  The recent progress of nickel-catalyzed asymmetric hydrofunctionalization of 1,3-dienes with different nucleophiles is reviewed by Long, Liu, Zhang, Zhu and Gu on page 3309. The substrate scope, limita-tions and mechanism characteristics of asymmetric hydrofunctionalization are dis-cussed. According to the different kinds of nucleophiles, it mainly includes asymmetric hydrocarbonation, asymmetric hydroamina-tion, asymmetric hydrophosphinylation and asymmetric hydroalkoxylation.
2024, 44(11)

25 November 2024
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REVIEW

Research Progress on Selective Multi-site Functionalization of Hydrocarbon Chains

Junwei Wang, Huikang Liu, Zehua Yang, Zhengxing Wu, Wanbin Zhang

Chinese Journal of Organic Chemistry 2024, 44 (11), pp 3273-3281 DOI: 10.6023/cjoc202404010

Abstract( 167) HTML( 8) PDF(632KB)( 234 )

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Research Progress in High-Performance Organic Small-Molecule Photovoltaic Donors Materials

Kaihuai Tu, Xue Jiang, Tainan Duan, Zeyun Xiao

Chinese Journal of Organic Chemistry 2024, 44 (11), pp 3282-3298 DOI: 10.6023/cjoc202403026

Abstract( 344) HTML( 0) PDF(1281KB)( 300 )

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Recent Progress on Fluorescent Probes for the Detection of Methylglyoxal

Yaping Wang, Yanling Fan, Yongqi Ren, Yulin Xu

Chinese Journal of Organic Chemistry 2024, 44 (11), pp 3299-3308 DOI: 10.6023/cjoc202403003

Abstract( 143) HTML( 4) PDF(664KB)( 148 )

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Recent Advances in Nickel-Catalyzed Asymmetric Hydrofunctionalization of 1,3-Dienes

Jiao Long, Baixue Liu, Shuangshuang Zhang, Yuanyuan Zhu, Shuangxi Gu

Chinese Journal of Organic Chemistry 2024, 44 (11), pp 3309-3320 DOI: 10.6023/cjoc202403021

Abstract( 226) HTML( 3) PDF(879KB)( 286 )

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Recent Progress on Methods for the Preparation of Mono/Di/Trifluoromethoxylation Reagents

Wei Zheng, Fengxue Liu, Hongqiong Zhao, Ying Xu, Ning Chen, Yingjie Liu

Chinese Journal of Organic Chemistry 2024, 44 (11), pp 3321-3334 DOI: 10.6023/cjoc202403011

Abstract( 196) HTML( 0) PDF(794KB)( 257 )

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Advances in Homogeneous Hydrogenation of Esters to Alcohols by Non-noble Metal Complexes

Xiaolong Fang, Yu Zhang, Tao Wang, Bin Li, Ning Duan, Fengjun Zhang

Chinese Journal of Organic Chemistry 2024, 44 (11), pp 3335-3344 DOI: 10.6023/cjoc202403024

Abstract( 156) HTML( 0) PDF(587KB)( 184 )

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Progresses in the Preparation of Chromone Compounds and Their Applications in Organic Synthesis

Zhonghao Li, Yu Zeng, Yong Zeng, Wenjin Xu, Xiying Cao, Yuting Guo, Qing Shen, Zhaoyang Wang

Chinese Journal of Organic Chemistry 2024, 44 (11), pp 3345-3356 DOI: 10.6023/cjoc202403025

Abstract( 283) HTML( 16) PDF(773KB)( 477 )

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ARTICLE

Design and Synthesis of Near-Infrared Fluorescent Dyes of Difluoroboron β-Diketonate and Cell Imaging

Yunpeng Qi, Wei Liu, Junlong Wang, Tao Du, Songlin Jiao

Chinese Journal of Organic Chemistry 2024, 44 (11), pp 3357-3364 DOI: 10.6023/cjoc202404032

Abstract( 88) HTML( 2) PDF(2820KB)( 89 )

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Synthesis of Multisubstituted 4H-Chromenes via Brønsted Base- Mediated Tandem Cyclization Reactions of β-(2-Hydroxyaryl) Ethenesulfonyl Fluorides and β,γ-Unsaturated Ketoesters (Ynones)

Delin Tang, Jinyun Luo, Guangfen Du, Zhihua Cai, Lin He

Chinese Journal of Organic Chemistry 2024, 44 (11), pp 3365-3374 DOI: 10.6023/cjoc202404037

Abstract( 109) HTML( 2) PDF(678KB)( 109 )

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Study on the Light Promoted One-Pot Three Component Aminoarylation Reaction of 1,4-Naphthoquinone

Bin Wang, Wancang Han, Yonghong Zhang, Yu Xia, Weiwei Jin, Ziren Chen, Shaofeng Wu, Chenjiang Liu

Chinese Journal of Organic Chemistry 2024, 44 (11), pp 3375-3385 DOI: 10.6023/cjoc202405001

Abstract( 92) HTML( 4) PDF(828KB)( 147 )

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Total Synthesis of trans-4'a-Methyl-3',4'a,9',10',10'a-hexahydro-spiro[cyclobutane-1,1'(2H)-phenanthrene]

Weihao Dai, Chenyu Huo, Tianlu Zheng, Daoyong Zhu, Shaohua Wang

Chinese Journal of Organic Chemistry 2024, 44 (11), pp 3386-3391 DOI: 10.6023/cjoc202404026

Abstract( 78) HTML( 3) PDF(516KB)( 79 )

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Se/ZrO₂-Catalyzed Oxidative Polymerization of Aniline

Daming Yong, Tingting Zuo, Qichao Wu, Xu Zhang

Chinese Journal of Organic Chemistry 2024, 44 (11), pp 3392-3398 DOI: 10.6023/cjoc202404022

Abstract( 92) HTML( 0) PDF(1552KB)( 174 )

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Preparation of Polyolefin Elastomers by Neutral Nickel Catalysts: Synergistic Effect of Steric Hindrance and Secondary Interaction

Qiankun Li, Hongliang Mu, Zhongbao Jian

Chinese Journal of Organic Chemistry 2024, 44 (11), pp 3399-3408 DOI: 10.6023/cjoc202403034

Abstract( 97) HTML( 1) PDF(2310KB)( 74 )

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Construction of 3,5-Diarylpyridine Derivatives Using N,N-Dimethyl-ethanolamine as a Single-Carbon Synthon

Xinyu Zhang, Jing Chen, Yongmin Ma

Chinese Journal of Organic Chemistry 2024, 44 (11), pp 3409-3416 DOI: 10.6023/cjoc202405008

Abstract( 82) HTML( 0) PDF(605KB)( 79 )

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A Turn-ON Near-Infrared Fluorescent Probe for the Detection of Dipeptidyl Peptidase IV Activity in Liver Cancers

Fei Zhang, Yu Mei, Xuefeng Ding, Zaifeng Li, Peng Zhang, Caifeng Ding

Chinese Journal of Organic Chemistry 2024, 44 (11), pp 3417-3426 DOI: 10.6023/cjoc202404028

Abstract( 118) HTML( 6) PDF(9132KB)( 125 )

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Copper-Catalyzed Synthesis of Benzofuropyrimidoisoindole Derivatives

Heng He, Lanlan Lü, Jianquan Liu, Xiangshan Wang

Chinese Journal of Organic Chemistry 2024, 44 (11), pp 3427-3436 DOI: 10.6023/cjoc202404005

Abstract( 107) HTML( 3) PDF(894KB)( 115 )

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Mechanochemistry Enabled Friedel-Crafts Alkylation Reactions of Donor-Acceptor Cyclopropanes with 2-Indolymethanols

Jinshao Liang, Lihong Ruan, Xurong Shi, Yinzhi Chen, Chuhuang Song, Jun'an Xiao, Zhiping Liu

Chinese Journal of Organic Chemistry 2024, 44 (11), pp 3437-3445 DOI: 10.6023/cjoc202404006

Abstract( 71) HTML( 0) PDF(700KB)( 141 )

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Design, Synthesis and Fungicidal and Nematocidal Activity of 1,2,3-Benzotriazine-4-one Oxadiazole Thioether (Sulfone) Methyl Derivatives

Wei Zhao, Fengyu Li, Wei Zhao, Run Zha, Caihua Shi, Zhihong Xu

Chinese Journal of Organic Chemistry 2024, 44 (11), pp 3446-3455 DOI: 10.6023/cjoc202403019

Abstract( 33) HTML( 1) PDF(2670KB)( 15 )

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Pd-Catalyzed Reductive Cross-Coupling of Allylic Esters with Aryl Iodides Involving the Insertion of SO₂

Xinwei Zhang, Shuizhen Lin, Xiaolei Huang

Chinese Journal of Organic Chemistry 2024, 44 (11), pp 3456-3466 DOI: 10.6023/cjoc202404019

Abstract( 87) HTML( 0) PDF(583KB)( 98 )

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Tetrahydroxydiboron and Copper Sulfate Co-Promoted Facile Synthesis of Phthalides

Feifei Fan, Longhui Chen, Guangwei Wang

Chinese Journal of Organic Chemistry 2024, 44 (11), pp 3467-3475 DOI: 10.6023/cjoc202405009

Abstract( 64) HTML( 0) PDF(1328KB)( 51 )

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Discovery of Alkyl Conjugated Diene Diacids as Novel ACLY Inhibitors

Tingting Cheng, Gaolei Song, Long Cheng, Fan Wang, Xinyu Sun, Zhifu Xie, Mei Zhang, Yangming Zhang, Jingya Li, Fajun Nan

Chinese Journal of Organic Chemistry 2024, 44 (11), pp 3476-3489 DOI: 10.6023/cjoc202405036

Abstract( 90) HTML( 3) PDF(4614KB)( 65 )

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Calcium Trifluoromethanesulfonimide Catalyzed Synthesis of 1-Substituted-amino-2-arylvinyl 1H-Indole-1-carboxylates

Yuying Zhang, Qingyan Song, Yuerong Li, Huaiji Zheng, Bangguo Wei

Chinese Journal of Organic Chemistry 2024, 44 (11), pp 3490-3496 DOI: 10.6023/cjoc202404007

Abstract( 87) HTML( 0) PDF(583KB)( 82 )

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Synthesis and Antitumor Activity of Novel Terephthalamide Derivatives

Yifei Gu, Caiju Wu, Siqi Wang, Shilin Zhang, Yuan Lu, Xinxin Si, Bailing Jiang

Chinese Journal of Organic Chemistry 2024, 44 (11), pp 3497-3504 DOI: 10.6023/cjoc202403049

Abstract( 86) HTML( 0) PDF(4572KB)( 100 )

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Rh(III)-Catalyzed Aminoalkylation of Alkenes with Diazo Compounds toward Functionalized Isoindolinones

Yuying Liu, Zhanwei Fu, Chao Yang, Mupeng Luo, Shurong Ban, Shouguo Wang

Chinese Journal of Organic Chemistry 2024, 44 (11), pp 3505-3517 DOI: 10.6023/cjoc202405016

Abstract( 177) HTML( 1) PDF(699KB)( 148 )

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Computational Insights into the Mechanism of the Mo-Catalyzed Deoxygenative Coupling of Aromatic Aldehydes

Qinghao Sun, Xiaoguang Bao

Chinese Journal of Organic Chemistry 2024, 44 (11), pp 3518-3525 DOI: 10.6023/cjoc202405018

Abstract( 98) HTML( 5) PDF(1043KB)( 130 )

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NOTE

Diterpenoids from Mangrove Plant Excoecaria agallocha L. and Their Anti-neuroinflammatory Activities

Junyi Li, Lu Yang, Mingbin Chen, Yong Rao, Zhongping Jiang, Ling Huang

Chinese Journal of Organic Chemistry 2024, 44 (11), pp 3526-3530 DOI: 10.6023/cjoc202404024

Abstract( 100) HTML( 0) PDF(1615KB)( 73 )

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Cu(OTf)₂ Catalyzed Rapid Nucleophilic Substitution of Propargyl Alcohols

Shunji Zhang, Huili Liu, Yun Jin

Chinese Journal of Organic Chemistry 2024, 44 (11), pp 3531-3540 DOI: 10.6023/cjoc202403050

Abstract( 103) HTML( 1) PDF(415KB)( 114 )

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Design, Synthesis and Antibacterial Activities of Osthole Derivatives Containing Thiazole Fragment

Jiaqiang Yang, Xuejiao Wu, Zicong Lu, Yangmi Chen, Huixian She, Haijun Liu

Chinese Journal of Organic Chemistry 2024, 44 (11), pp 3541-3549 DOI: 10.6023/cjoc202404030

Abstract( 128) HTML( 0) PDF(854KB)( 86 )

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Convergent Strategy to Synthesize (S)-8-(4-((1-(3-Fluoropropyl)-pyrrolidin-3-yl)oxy)phenyl)-7-(4-hydroxyphenyl)-5,6-dihydronaphthalen-2-ol as a Selective Estrogen Receptor Degrader

Panpan Chen, Xiaowei Feng, Zhipeng Lu, Tingyou Li

Chinese Journal of Organic Chemistry 2024, 44 (11), pp 3550-3555 DOI: 10.6023/cjoc202403009

Abstract( 122) HTML( 1) PDF(401KB)( 66 )

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Palladium-Catalyzed Synthesis of 2-(1-Isochromen-3-yl)acetalde-hydes via Carboxyl-Directed C(sp²)—H Alkylation/Annulation

Yue Wang, Xuyan Yang, Tianyu Liu, Tuanjie Li, Kai Zhang, Changsheng Yao

Chinese Journal of Organic Chemistry 2024, 44 (11), pp 3556-3563 DOI: 10.6023/cjoc202410013

Abstract( 40) HTML( 0) PDF(587KB)( 20 )

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HIGHLIGHT

Synthesis of Bridged Five-Membered Ring Systems by Type II [3＋2] Annulation of Allenylsilane-Ene

Tao Xu

Chinese Journal of Organic Chemistry 2024, 44 (11), pp 3564-3565 DOI: 10.6023/cjoc202400055

Abstract( 31) HTML( 3) PDF(411KB)( 17 )

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Bifunctional Chiral Electrocatalysts Enable Enantioselective α-Alkylation of Aldehydes

Jiayin Zhang, Chang Guo

Chinese Journal of Organic Chemistry 2024, 44 (11), pp 3566-3567 DOI: 10.6023/cjoc202400056

Abstract( 25) HTML( 2) PDF(436KB)( 20 )

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From Single-Electron Reduction to Single-Electron Oxidation: A New Strategy for Radical Coupling of Aldehyde and Olefins

Junwei Shi, Liangqiu Lu

Chinese Journal of Organic Chemistry 2024, 44 (11), pp 3568-3570 DOI: 10.6023/cjoc202400057

Abstract( 40) HTML( 4) PDF(395KB)( 39 )

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Visible-Light-Driven Multicomponent Reactions for the Versatile Synthesis of Thioamides by Radical Thiocarbamoylation

Qilong Wu, Daoshan Yang

Chinese Journal of Organic Chemistry 2024, 44 (11), pp 3571-3573 DOI: 10.6023/cjoc202400058

Abstract( 48) HTML( 4) PDF(428KB)( 46 )

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