Chinese Journal of Organic Chemistry 2026, 46(1)

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- About the Cover:
  
  13 new thiochromone formamide derivatives substituted at position 2 were synthesized and two synthetic routes for these compounds were developed by Zhou, Su, Cui, Cheng, Li, Zhou, Sun, and Li on page 87. Their antifungal activities against Gaeumannomyces graminis/ var. tritici were evaluated in vitro by the plate method. The results of structure-activity relationship indicated that the group at position 2 of thiochromone formamide derivatives had an important influence on their antifungal activities against Gaeumannomyces graminis var. tritici.
- About the Cover:
  
  The nickel-catalyzed borylation of aryl nonaflates with B2pin2 is reported by Liang, Gui, Wang, Chu, Xu, and Shen on page 207. The reactions proceeded effectively via C—O bond cleavage to afford various valuable arylboronates in moderate to excellent yields with good functionality tolerance. Additionally, gram-scale synthesis and late-stage functionalization of aryl nonaflate derived from pterostilbene could also be realized.
2026, 46(1)

25 January 2026
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REVIEWS ARTICLES HIGHLIGHTS

REVIEWS

Recent Advances on the Functionalization of Azlactones at Different Reactive Sites

Jiang Zhijie, Chen Jinxiu, Zhu Xiaofei, Deng Xinhao, Yan Qiongjiao, Wang Wei, Zhou Hui

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 1-20 DOI: 10.6023/cjoc202506007

Abstract( 73) HTML( 0) PDF(1112KB)( 28 )

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Recent Progress in the Total Synthesis of abeo-Steroids

Zhao Lilin, Li Zhaoqi, Zhong Liping, Min Long

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 21-38 DOI: 10.6023/cjoc202506022

Abstract( 146) HTML( 0) PDF(999KB)( 57 )

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Structural Modifications, Structure-Activity Relationships, and Total Synthesis Advances in Erythromycin Analogs against Resistant Pathogens

Cui Xinyi, Guo Lifan, Ma Congxuan, Li Yun, Liang Jianhua

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 39-73 DOI: 10.6023/cjoc202506020

Abstract( 56) HTML( 0) PDF(2154KB)( 22 )

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Progress in the Synthesis and Biological Studies of S-1-Propenyl-L-cysteine from Garlic

Tian Lingyan, Wang Shoufeng, Zeng Wei

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 74-86 DOI: 10.6023/cjoc202505028

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ARTICLES

Synthesis of Thiochromone Formamide Derivatives and Their Antifungal Activities

Zhou Pu, Su Ziyang, Cui Deyun, Cheng Yi-Nan, Li Yi, Zhou Haifeng, Sun Bingjian, Li Honglian

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 87-95 DOI: 10.6023/cjoc202506027

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Study on the Cyclopropanation Reactivity and Selectivity of Spiroannulated Pentacyclic Diastereoisomers toward Synthesizing Cryptoquinonemethides

Zhang Yuanhe, Shen Yunjie, Tan Dongxing, Han Fushe

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 96-105 DOI: 10.6023/cjoc202508010

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Study on the Synthesis and Fungicidal Activity of 1-Azolyl-1,1- diarylmethanes Containing Pyridine Ring

Hong Sai, Yin Fahong, Chen Minghui, Fu Bin, Xiao Yumei, Qin Zhaohai

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 106-117 DOI: 10.6023/cjoc202506035

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Silver-Catalyzed Tandem Decarboxylative Cyclization of 2,2-Difluoro-2-(phenylthio)acetic Acids with 2-Aryl-N-acrylamide Indoles

Liu Jiale, Tang Yucai, Yin Qiumei, Huang Jiaming, Deng Shiqiang, Xia Weiming, Jiang Jie, Wang Zu-Li

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 118-127 DOI: 10.6023/cjoc202507011

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Synthesis and Characterization of Silacyclopropenes

Chen Yilin, Yue Jiayi, Lin Yiming, Liu Bingni, Dai Wen, Zhu Hongping

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 128-134 DOI: 10.6023/cjoc202506023

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Visible-Light-Driven Halogen-Bond-Induced Direct Coupling of Diethyl α-Iodomethylphosphonates with Coumarins/Quinolinones

Liang Jiarui, Li Jinlan, Jiang Yun, Yao Qiuli, Xu Yingshu, Wang Anjun

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 135-145 DOI: 10.6023/cjoc202506016

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Regio-reversed [3＋2] Cycloaddition of Triketone Enones with Nitrones

Han Tianjiao, Shi Qianqian, Fu Yundong, Mei Guangjian

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 146-155 DOI: 10.6023/cjoc202507022

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Heterogeneous Copper Catalyzed Aerobic Oxidative Cross-Coupling of Tertiary Amines with Alkynes

Tan Ziyun, Yang Xin, Gong Shaofeng, Yang Huiling, Xie Yongyan, Zhang Jingya, Feng Zhetai, Li Wenyi, Xiao Xinsheng

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 156-166 DOI: 10.6023/cjoc202504020

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Copper-Catalyzed Asymmetric Oxidative Homocoupling Reaction of 3-Hydroxy-2-naphthoates: Design and Optimization of Amino Acid-Based Ligands

Wang Wen-Long, Wen Jia-Xu, Chen Fei, Bo Chunbo, Li Min, Liu Ning, Du Zhi-Hong

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 167-180 DOI: 10.6023/cjoc202505013

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Four-Component Hydroxythiolation of Styrenes with Imidazopyridines and Potassium Thiocyanate

Wang Yu, Huang Hongkun, Ling Chun, Chen Tian, Yao Hua, Yan Zhaohua

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 181-188 DOI: 10.6023/cjoc202506001

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S-Heteroarylation of Cysteines

Zhang Xin, Li Fei, Zhou Chenxing, Huo Congde

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 189-198 DOI: 10.6023/cjoc202506011

Abstract( 95) HTML( 0) PDF(607KB)( 41 )

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Study on FeCl₃-Mediated Reaction of Aryl Boronic Esters with Electrophiles

Cui Lihua, Li Yatong, Wang Qifeng

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 199-206 DOI: 10.6023/cjoc202506018

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Nickel-Catalyzed Borylation of Aryl Nonaflates for the Efficient Synthesis of Arylboronates via C—O Bond Functionalization

Liang Yuan, Gui Chao, Wang Wenwen, Chu Xueqiang, Xu Hao, Shen Zhiliang

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 207-214 DOI: 10.6023/cjoc202507010

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Photocatalytic Radical-Mediated Synthesis of Unnatural α-Amino Acids from Heteroaryl Aldehydes

Ren Ke, Zhang Guanglu, Niu Yifan, Wang Xiaomeng, Chen Canyu, Jiang Min

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 215-224 DOI: 10.6023/cjoc202507030

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PPh₃-Mediated One-Pot Synthesis of Indolin-3-ones from 2-Alkynylnitrobenzenes and Indoles

Feng Faxiu, Xu Shijie, Wang Xue, Yang Zhuoran, Wang Wenjun, Huang Shenlin, Zhang Xiaoxiang

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 225-232 DOI: 10.6023/cjoc202506013

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Schiff Base Type Fe(III) Complexes Catalyzed Carbon Dioxide and Epoxides for Preparing Cyclic Carbonates

Liu Tao, Zhou Yongbo, Lang Tongqing, Niu Haibo, Chen Fei, Du Zhihong, Bo Chunbo, Li Min, Liu Ning

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 233-240 DOI: 10.6023/cjoc202506003

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Efficient Hydrogenation of Ketones to Alcohols Catalysed by Phosphinoamine Rhenium Complexes

Fang Xiaolong, Wang Jun, Xu Shuting, Li Hao, Hu Kun, Chen, Yiyu

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 241-249 DOI: 10.6023/cjoc202506024

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Design, Synthesis and Anticancer Activity Evaluation of Novel Nitrogen-Containing Heterocyclic Compounds Based on Nitidine Skeleton

Su Xiaowei, Xu Hao, Zhou Huafeng, Wang Xiajie, Li Peiyuan, Xia Xing, Chen Wenya, Huo Lini

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 250-265 DOI: 10.6023/cjoc202504032

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Nickel/Visible Light Dual-Catalyzed C—O Bond Coupling Reactions of Aryl Bromides with Alcohols

Gao Shan, Xie Xin, Liu Yuanhong

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 266-278 DOI: 10.6023/cjoc202506009

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Synthesis of α,β-Disubstituted Acrylates via PPh₃-Catalyzed Ring-Opening Addition Reaction of Cyclopropenones with Alkyl Bromides at Room Temperature

Xu Cheng, Peng Tao, Zhou Mengyuan, Liu Minglin, Huang Xiaoqing, Wang Yongfeng, Liu Zheng, Yin Guodong

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 279-288 DOI: 10.6023/cjoc202505033

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Characterization of Glutarimide Derivatives from Agrimonia pilosa-Associated Endophytic Streptomyces sp. YINM00048

Su Yuying, Wang Yingfang, Yi Mengzhuo, Zhao Lixing, Li Jiaxuan, Ma Ling, Yin Min

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 289-294 DOI: 10.6023/cjoc202506015

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Activation of the Biosynthetic Gene Cluster in Streptomyces sp. YINM00050 Facilitated the Discovery of a Novel Benzoisochromanequinone

Zhang Yuan, Guo Ying, Yang Mingxi, Dong Kui, Zhao Lixing, Ma Ling, Yin Min

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 295-299 DOI: 10.6023/cjoc202506021

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Two New Linear Furocoumarins from Notopterygium incisum and Their Anti-inflammatory Activity

Hu Su, Zhao Lilian, Li Xinyu, Ye Yubei, Deng Yun, Huang Lijun, Guo Dale

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 300-303 DOI: 10.6023/cjoc202505002

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HIGHLIGHTS

Chiral Bicyclic Imidazole-Catalyzed Phosphorus Atom Activation and Asymmetric Construction of Diverse P(V) Compounds

Wu Xiuli, Wu Xingxing

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 304-305 DOI: 10.6023/cjoc202600001

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Chiral Octahedral Cobalt(III)-Catalyzed C—H Macrocyclization to Access Planar-Chiral Cyclophanes

Wen Yilu, Zhao Changgui

Chinese Journal of Organic Chemistry 2026, 46 (1), pp 306-307 DOI: 10.6023/cjoc202600002

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