Chinese Journal of Organic Chemistry 2021, 41(2)

- About the Cover:
  
  Enantioselective electrophilic thiolation of alkenes has emerged as a straightforward pathway for the synthesis of chiral sulfides. By this fashion, both the thio group and another valuable functional group can be introduced sim-ultaneously into the parent alkene molecules. This account focuses on the advance on chiral bifunctional chalcogenide-catalyzed enantioselective electrophilic thiofunctionalization of alkenes, which is reported by Jiang and Zhao on page 443.
- About the Cover:
  
  Fe-catalyzed borylation of ketones to access tertiary α-hydroxyboronates has been demonstrated by Zhu, Xia, and Liu on page 661. In this transformation, commercially available FeBr2 was used as the catalyst, various aliphatic ketones with different functional groups or steric hinderance have been converted into tertiary α-hydroxyboronates efficiently.
2021, 41(2)

25 February 2021
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ACCOUNT

Chiral Bifunctional Chalcogenide-Catalyzed Enantioselective Electrophilic Thiofunctionalization of Alkenes

Quanbin Jiang, Xiaodan Zhao

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 443-454 DOI: 10.6023/cjoc202010005

Abstract( 1751) HTML( 60) PDF(858KB)( 1834 )

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Review

Recent Progress in Aryne Participated Dearomatization Reactions

Qiang Yan, Rong Fan, Binbin Liu, Shuaisong Su, Bo Wang, Tuanli Yao, Jiajing Tan

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 455-470 DOI: 10.6023/cjoc202009009

Abstract( 1640) HTML( 57) PDF(1018KB)( 1898 )

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Recent Progress in Catalytic Asymmetric Alkynylation of Imines

Shurui Zhou, Kaige Wen, Xingping Zeng

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 471-489 DOI: 10.6023/cjoc202007043

Abstract( 1294) HTML( 53) PDF(985KB)( 2120 )

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Research and Application of 2-Iodoxybenzoic Acid in Organic Synthesis

Shuyu Zhang, Haotian Wu, E Tang

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 490-503 DOI: 10.6023/cjoc202007030

Abstract( 1112) HTML( 34) PDF(846KB)( 1624 )

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Advances in Fluorinated Organometallic Complexes with Aggregation-Induced Emission Characteristics

Chengyuan Qin, Jinling Miao, Yong Nie, Wei Liu, Ying Gao, Tianrui Li, Xuchuan Jiang

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 504-520 DOI: 10.6023/cjoc202007015

Abstract( 899) HTML( 26) PDF(3006KB)( 1272 )

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Progress in Annulative Transformations from Indoles to Carbazoles: State of the Art

Yuying Du, Yeyuan Xiao, Fuli Tian, Limin Han, Yanlong Gu, Ning Zhu

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 521-528 DOI: 10.6023/cjoc202007014

Abstract( 1262) HTML( 106) PDF(641KB)( 1345 )

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Recent Advances in Cross-Dehydrogenative-Coupling Reactions Using Molecular Oxygen as the Sole Oxidant

Weihui Zhuang, Xiaofeng Zhang, Qiufeng Huang

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 529-542 DOI: 10.6023/cjoc202007007

Abstract( 1109) HTML( 34) PDF(998KB)( 1375 )

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Recent Advances in C—H Fluorination and Amination with N-Fluorobenzenesulfonimide

Weilin Wang, Weidong Chen, Junfei Luo, Pan Xie

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 543-552 DOI: 10.6023/cjoc202006069

Abstract( 993) HTML( 39) PDF(699KB)( 1792 )

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Progress in Biological Activity and Synthesis of Nematode Hatching Pheromone Glycinoeclepin A

Ding Ma, Junli Ao, Naifeng Hu, Guangxin Liang

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 553-566 DOI: 10.6023/cjoc202006065

Abstract( 964) HTML( 13) PDF(870KB)( 1464 )

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Application of Boronate Bond in Drug Delivery System

Lijuan Wang, Xianliang Sheng, Jie Wang, Yuhui Zhang

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 567-581 DOI: 10.6023/cjoc202006060

Abstract( 2427) HTML( 96) PDF(4383KB)( 2630 )

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REVIEW

Application of Cascade Reactions in the Synthesis of Sprio-hetero- cycles Initiated by Intramolecular Cyclization of Alkynols

Shuyan Yu, Lihong Gao, Yizhe Yan, Zhigang Yin, Yongjia Shang

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 582-593 DOI: 10.6023/cjoc202006050

Abstract( 836) HTML( 14) PDF(739KB)( 988 )

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Review

Progress in the Synthesis of Pyrrole-2-carboxylate Catalyzed by Transition Metals

Ci Li, Mingrui Li, Yuxing Xie, Yang Yu, Fei Huang

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 594-610 DOI: 10.6023/cjoc202006048

Abstract( 823) HTML( 13) PDF(1096KB)( 1002 )

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Recent Advances in Fluorescent Probes for Biothiols

Li Chen, Junbo Li, Dugang Chen

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 611-623 DOI: 10.6023/cjoc202006046

Abstract( 2907) HTML( 109) PDF(1029KB)( 2343 )

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Synthesis of Novel Porous Organic Materials Based on Phloroglucinol and Its Derivatives

Hanlin Deng, Xiansheng Luo, Zhihua Li, Jiangying Zhao, Muhua Huang

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 624-641 DOI: 10.6023/cjoc202005070

Abstract( 1284) HTML( 59) PDF(2160KB)( 1512 )

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Application of α-Aminoalkyl Radical in Visible Light Catalysis

He Zhao, Dongping Cheng, Xiaoliang Xu

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 642-660 DOI: 10.6023/cjoc202005055

Abstract( 1374) HTML( 41) PDF(1110KB)( 1586 )

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Article

Iron-Catalyzed Borylation of Ketones to α-Hydroxyboronates

Qing Zhu, Chungu Xia, Chao Liu

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 661-668 DOI: 10.6023/cjoc202010022

Abstract( 1275) HTML( 35) PDF(499KB)( 1480 )

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Ag-Catalyzed Reactions of 3-Trifluoroacetyl Indoles and Isocyano- acetates: An Efficient Process to (Z)-β-Trifluoromethylated Dehydrotryptophan Derivatives

Mingliang Zhang, Pin Zhao, Hao Yuan, An'an Zhang, Wenyu Zhang, Linlin Zheng, Dongqing Wu, Lantao Liu

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 669-676 DOI: 10.6023/cjoc202008023

Abstract( 896) HTML( 14) PDF(716KB)( 802 )

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Synthesis of Multi-substituted 1,4-Dihydroquinoline Derivatives from Morita-Baylis-Hillman (MBH) Carbonates

Hongyan Shi, Ying Zhong, Zhigang Zhao

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 677-687 DOI: 10.6023/cjoc202008020

Abstract( 989) HTML( 20) PDF(720KB)( 946 )

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Cyanuric Chloride Catalysis and Solvent Effect Leading to a Mild and Efficient Beckmann Rearrangement of Ketoximes

Tingting Zhou, Xia Liu, Zihang Ye, Yipeng Zhou, Yaqi Yang, Qing Xu

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 688-694 DOI: 10.6023/cjoc202008018

Abstract( 762) HTML( 27) PDF(558KB)( 1398 )

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Study on the Copper-Catalyzed Selective Allylation of Aryl (or Alkyl) Halides

Boshi Han, Zheng Shi, Huihong He, Xinghua Zhang

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 695-701 DOI: 10.6023/cjoc202008012

Abstract( 768) HTML( 13) PDF(494KB)( 911 )

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Microwave-Assisted Synthesis of Perylene Monoimide Derivatives

Ya'nan Wang, Chong Wang, Yuming Qi, Guokai Li, Xiaoliu Li, Kerang Wang

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 702-707 DOI: 10.6023/cjoc202008010

Abstract( 779) HTML( 19) PDF(497KB)( 735 )

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Design, Synthesis and Biological Activities of Myricetin Derivatives Containing Quinazoline Thioether Moiety

Jun He, Xuemei Tang, Qing Zhou, Feng Peng, Tingting Liu, Liwei Liu, Ming He, Chengwei Xie, Wei Xue

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 708-718 DOI: 10.6023/cjoc202008006

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A Naphthalimide-Based Hypochlorous Acid-Selective Fluorescent Probe and Its Application in Cell Imaging

Xinyu Wang, Shaolong Qi, Jianshi Du, Qiang Li, Lubao Zhu, Longqi Xue, Qing Zhao, Qingbiao Yang, Yaoxian Li, Xianling Cong

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 719-725 DOI: 10.6023/cjoc202008005

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Synthesis of the ABC Ring System of Wallichanol Natural Product

Gang Yang, Xiangyu Feng, Congcong Han, Yang Chen, Shuzhong He

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 726-730 DOI: 10.6023/cjoc202008001

Abstract( 694) HTML( 20) PDF(509KB)( 985 )

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Synthesis of 2-Quinolinone Derivatives via [3+3] Cyclization Promoted by Acetic Anhydride

Yu Zhao, Zhuo Chen, Xuebing Chen

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 731-737 DOI: 10.6023/cjoc202007070

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Synthesis and Antimicrobial Activities of Novel 1,3,4-Oxa(Thia)- diazole Derivatives Containing 6-Fluoroquinazoline Moiety

Jun Shi, Na Luo, Muhan Ding, Chuanhui Li, Suran Wan, Peijia Li, Junhong Li, Xiaoping Bao

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 738-756 DOI: 10.6023/cjoc202007068

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Access to Tetrasubstituted Tri(indolyl)methanes through Copper-Catalyzed Addition/Substitution Sequence

Wenbo Wang, Huabin Han, Lele Wang, Qilin Wang, Zhanwei Bu

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 757-765 DOI: 10.6023/cjoc202007055

Abstract( 603) HTML( 9) PDF(778KB)( 636 )

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Synthesis of Alkynes Composed of the Novel Substituents and Their Reactions with B(C₆F₅)₃

Xin Xi, Gongping Zhang, Jiancheng Li, Yanting Huang, Wenjun Jiang, Peng Wu, Hongping Zhu

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 766-775 DOI: 10.6023/cjoc202007018

Abstract( 654) HTML( 5) PDF(1159KB)( 557 )

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Synthesis and Antitumor Activity of Novel Pyrimidine Monocyclic Nonclassical Antifolates

Jing Cong, Fang Fang, Liangmin Xue, Meng Wang, Chao Tian, Xiaowei Wang, Junyi Liu, Zhili Zhang

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 776-787 DOI: 10.6023/cjoc202007006

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Synthesis of Stable Isotope Labeled ¹³C₄-1,4-Dihydropyridines on 5,6-Position and Its Substituent Carbon

Yuzhao Hu, Haiyuan Quan, Liuyang Wang, Zhinan Wang, Xiangdong Mei, Jun Nin, Dongmei She

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 788-794 DOI: 10.6023/cjoc202006078

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Nucleophilic Etherification of Heteroaryl Alkyl Ethers, Heteroaryl Halides with (Deuterated) Alcohols

Xia Wang, Yixin Qu, Chengyu Long, Xue-Qiang Wang

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 795-805 DOI: 10.6023/cjoc202006077

Abstract( 798) HTML( 13) PDF(535KB)( 770 )

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One-Pot Synthesis of 1,5-Benzodiazepine Compounds by Three-Component Tadem Reaction

Jing Li, Zhenfang Hao, Kaiyue Zhang, Lanzhi Wang

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 806-818 DOI: 10.6023/cjoc202006040

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One-Pot Three-Component Synthesis of Novel 1,5-Benzodiazepine Derivatives and Their anti-BVDV (Bovine Viral Diarrhea Virus) Activity

Chao Han, Lei Nie, Xiao Han, Yan Zhang, Kelei Sun, Lei Shi, Guanghua Cui, Wei Meng

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 819-825 DOI: 10.6023/202004018

Abstract( 593) HTML( 9) PDF(632KB)( 474 )

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NOTE

Synthesis and Fungicidal Activity of Novel Allyl Benzoate Compounds Containing Triazole

Wei Yu, Han Wang, Li-Jing Min, Xue-Wen Hua, Xing-Hai Liu

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 826-832 DOI: 10.6023/cjoc202006037

Abstract( 526) HTML( 19) PDF(1509KB)( 939 )

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Visible-Light-Induced Preparation of Quinazolinones by Oxidation of Benzyl Alcohols in Water

Fan Zhang, Huiqing Hou, Xiuzhi Xu, Zhitao Chen, Fang Ke

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 833-841 DOI: 10.6023/cjoc202007027

Abstract( 788) HTML( 16) PDF(754KB)( 885 )

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Design, Synthesis and Fungicidal Activities of Pyridyl Oxazoamide Compounds

Shu Chen, Chaoli Ren, Xiaoyu Tian, Donglin Zhang, Sen Yang, Shaoqing Yuan, Xiaohua Du, Chengxia Tan

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 842-848 DOI: 10.6023/cjoc202007009

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Palladium-Catalyzed Stereoselective 1,3-Diarylation of 1,4-Cyclohexadiene

Hailiang Pang, Dong Wu, Guoyin Yin

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 849-856 DOI: 10.6023/cjoc202006022

Abstract( 938) HTML( 17) PDF(519KB)( 936 )

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HIGHLIGHT

Asymmetric Formal Hetero-Ene Reaction of Allylgold Intermediates

Weidi Cao, Xiaohua Liu

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 857-858 DOI: 10.6023/cjoc202100009

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Electrochemical 1,2-Diarylation of Alkenes Enabled by Direct Dual C—H Functionalizations of Electron-Rich Aromatic Hydrocarbons

Ziqiang Wang, Chen Zhu

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 859-860 DOI: 10.6023/cjoc202100010

Abstract( 628) HTML( 21) PDF(400KB)( 707 )

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Nickel-Catalyzed Four-Component Carbocarbonylation of Alkenes under Atmospheric CO

Binqing He, Xuesong Wu

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 861-862 DOI: 10.6023/cjoc202100011

Abstract( 526) HTML( 12) PDF(376KB)( 813 )

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Enantioselective Alkylation of Azoles by Merging Visible Light and Copper Catalysis

Xiangsheng Li, Qiang Liu

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 863-864 DOI: 10.6023/cjoc202100012

Abstract( 499) HTML( 13) PDF(384KB)( 643 )

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Palladium-Catalyzed Asymmetric Markovnikov Hydroaminocarbonylation of Alkenes

Duanshuai Tian, Wenjun Tang

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 865-866 DOI: 10.6023/cjoc202100013

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Carbamoyl Fluoride-Promoted Ni-Catalyzed Asymmetric Carbamoyl-Arylation of Unactivated Alkenes

Xianqing Wu, Yifeng Chen

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 867-868 DOI: 10.6023/cjoc202100014

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Regioselective Markovnikov Hydrodifluoroalkylation of Difluoroenoxysilanes with Alkenes

Guoshu Chen, Yunlin Liu

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 869-870 DOI: 10.6023/cjoc202100015

Abstract( 519) HTML( 11) PDF(431KB)( 550 )

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Visible-Light-Driven Sulfonamide Catalyzed Alkylation of α-C(³)—H Bonds of Heteroatoms

Quanqing Zhao, Jiarong Chen

Chinese Journal of Organic Chemistry 2021, 41 (2), pp 871-872 DOI: 10.6023/cjoc202100016

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