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About the Cover:A series of novel N-2,3-difluorophenyl cyclobu-tylamine M4 AChR positive allosteric modulators were designed and synthesized by Liu, Chen, Tian, Zhou, Zhou and Liu on page 2138. The assays on M4 receptor cells showed that some target compounds displayed activities higher than or comparable to the lead compound, providing a guidance for developing new M4 AChR positive allosteric modulators.
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